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3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-(2-methylpropyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-methylbut-2-en-1-one
4-(3-hydroxy-3-methylbutyl)-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}benzamide
4-[2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3-thiazol-2-amine
3-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-4H-chromen-4-one
methyl(pyridin-2-ylmethyl)[1-(pyridin-3-yl)propyl]amine
3-[3-(dimethylamino)propyl]-8-methyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-propyl-2-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
2-methyl-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-amino-6-(4-methoxyphenyl)-4-[2-(methylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
7-[(2-fluorophenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-tert-butyl-4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
10-methoxy-5-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
5-(4-methoxyphenyl)-N-[5-(morpholin-4-yl)pentyl]-1,2,4-triazin-3-amine
2-[cyclohexyl(methyl)amino]-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)pyridine-3-carboxamide
2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-(4-methoxyphenyl)acetic acid
N-cyclopropyl-1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
2-[5-cyclopropyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
N-(2,3-dihydro-1H-inden-2-yl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-propylacetamide
4-ethyl-1-methyl-3-{[1-(3-methylbenzenesulfonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-(cyclohexylmethyl)-N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-ol
3-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}piperidine-1-carboxamide
4-[2-(1-phenyl-1H-1,2,4-triazol-5-yl)phenyl]-1λ6-thiomorpholine-1,1-dione
1'-(isoquinoline-5-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[4-(2,5-dimethoxybenzoyl)benzoyl]-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
(1R,5S,6S)-3-cyclopentyl-6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-3-azabicyclo[3.1.0]hexane
N-[(3S,5S)-5-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}-1-methylpyrrolidin-3-yl]thiophene-2-carboxamide
2-(2-{[2-(5-methylthiophen-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[4-(3,6-dimethylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane
N,N-diethyl-1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-4-carboxamide
2-[(2,6-dichlorophenyl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{3-[2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
3-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-4-(3-methylpiperidin-1-yl)benzamide
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-(pyrrolidin-1-yl)pyrrolidine
1-[(2,4-dimethoxyphenyl)methyl]-4-phenoxypiperidine-4-carboxylic acid
1-{3-[2-(cyclohexylmethyl)morpholin-4-yl]-3-oxopropyl}azepan-2-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-(oxolan-2-yl)-N-(propan-2-yl)thiophene-2-carboxamide
3-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
4-[(2-fluorophenyl)methyl]-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
1-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
2-(1-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
2-(furan-2-yl)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(1H-indol-4-yl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one