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3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-dihydroquinoxalin-2-one
2-[(2S)-2-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]-3-phenylpropanamido]acetic acid
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]methanesulfonamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-methyl-1,3,4-oxadiazol-2-amine
6-{[(1R,5S)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
1-[(4aR,8aR)-4a-hydroxy-7-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-cycloheptyl-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
(2R)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(methoxymethyl)pyrrolidine
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-benzyl-8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
6-[2-(piperidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-4-methoxyphenol
methyl 2-[3-oxo-1-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-yl]acetate
8-(1-benzofuran-5-ylmethyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(3,4-difluorophenyl)-1-(quinoxaline-6-carbonyl)piperidin-3-amine
N-cyclopropyl-1-[3-(1H-indol-3-yl)propanoyl]piperazine-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-2-(4-propanoylphenoxy)acetamide
N2-{[2-(1H-imidazol-1-yl)phenyl]methyl}-N4,N4,5-trimethylpyrimidine-2,4-diamine
1-tert-butyl-4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
3-methyl-N-{2-[1-(pyridin-3-ylmethyl)piperidin-3-yl]ethyl}pyridine-4-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidine-2-carboxamide
N-butyl-2-[1-(2-fluoro-5-sulfamoylphenyl)-N-methylformamido]acetamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-4-yl]pyridine-2-carboxamide
5-methoxy-1,2-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-indole-3-carboxamide
5-(azocan-1-yl)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)propanamide
3-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}-4H-chromen-4-one
1-(oxan-4-yl)-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
N4-[(4,6-dimethylpyridin-2-yl)methyl]-5-ethyl-N4-methylpyrimidine-2,4-diamine
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-(pyridin-4-ylsulfanyl)acetamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(3-hydroxy-3-methylbutyl)benzamide
12-(azepane-1-carbonyl)-5-chloro-15-methyl-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
2-{2-[(dimethylamino)methyl]-4-(pyridin-3-yl)phenoxy}-N-(furan-2-ylmethyl)acetamide
N-cyclopropyl-2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}pyridine-4-carboxamide
methyl N-{[(2S,4S)-4-fluoro-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)pyrrolidin-2-yl]methyl}carbamate
2-(morpholin-4-yl)-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-4-amine
2-[(2-fluorophenyl)methyl]-4-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-ethyl-2,4-dimethyl-N-(pyridin-4-ylmethyl)-1,3-oxazole-5-carboxamide
2-methoxy-5-(4-phenyl-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-5-yl)phenol
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(pyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
5-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3,5-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
3-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-4-yl)benzonitrile
2-hydroxy-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-benzyl-N-methylpropanamide