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N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1,3-benzothiazole-6-carboxamide
{imidazo[1,2-a]pyrimidin-6-ylmethyl}(2-methoxyethyl)[(4-methylphenyl)methyl]amine
methyl 2-(3-{[3-(phenylamino)piperidin-1-yl]methyl}-1H-indol-1-yl)acetate
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
N-(2-fluorophenyl)-4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-benzyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]pyrrolidin-3-amine
1-[1-(methoxymethyl)cyclopentyl]-3-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]urea
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]piperidin-2-one
2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-{[(1-ethylpiperidin-4-yl)amino]methyl}-2-methylpyrrolidin-2-yl]methanol
3,5-dimethyl-4-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
5-ethyl-2,3-dimethyl-N-[2-(pyrazin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{[3-(furan-2-yl)-1-methyl-1H-1,2,4-triazol-5-yl]methyl}-4-phenylpyrrolidin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(pyridin-3-yl)acetamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(3-methoxy-4-methylbenzoyl)piperidin-3-yl]propanamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(methylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperazin-2-one
5-({2-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1-methyl-1H-1,2,3,4-tetrazole
6-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(methylsulfanyl)propan-1-one
methyl 3-[2-(2-fluorophenyl)acetyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5S,6S)-6-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
4-(benzyloxy)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
[1-(1H-1,3-benzodiazol-2-ylmethyl)-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl]methanol
2-(2,2-dimethyloxan-4-yl)-4-{3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-ethyl-5-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-4-sulfonamide
[(8-methoxyquinolin-2-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
2-(furan-2-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]azepane
(1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
(4aS,8aR)-2-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-decahydroisoquinoline
(3S,4S)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
7-{2-[(dimethyl-1H-1,2,4-triazol-1-yl)methyl]propanoyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{4-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}pyridine
3-(2-fluorophenoxymethyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
(4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1,4-oxazepan-6-yl)methanol
1-{3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}imidazolidin-2-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
2-cyclohexyl-5-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}pyrimidine
N-(3-fluoro-2-methylphenyl)-2-{[1-(4-fluorophenyl)-2-methylpropan-2-yl]amino}acetamide
N-(4-fluoro-2-methylphenyl)-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]propanamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-methyl-1H-imidazole-5-carboxamide
6,8-dimethyl-3-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]-1,2-dihydroquinolin-2-one
2-(5-acetylthiophen-3-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propyl-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
7-cyclohexyl-2-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2,3-difluoro-6-methoxy-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-(4-methylpiperidin-1-yl)-3-[(1,2,3,4-tetrahydronaphthalen-2-yl)amino]propan-1-one