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5-{1-[3-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
1-(3-benzoylpiperidin-1-yl)-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
3-(2,4-dimethoxyphenyl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(4-hydroxyphenyl)propan-1-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
N'-cyclopentyl-N'-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-N,N-dimethylbutanediamide
5-[(1-benzothiophen-2-ylmethyl)(methyl)amino]-1-benzyl-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(1S,5R)-6-(4-chloro-2-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-(3-methoxypropyl)-3-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(morpholin-4-yl)-2-[(2-phenylphenyl)methyl]-2,3-dihydropyridazin-3-one
2-ethoxy-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
2-{[4-(2-methoxyphenyl)-5-(1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
9-(5-ethylpyrimidin-2-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-[(1-methylpyrrolidin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(thiophen-3-yl)ethan-1-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-ethyl-4-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-indole
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-3-methoxypropanamide
N-[2-(azepan-1-yl)-2-phenylethyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
4-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)benzonitrile
2-(4-chlorophenyl)-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]morpholine
2-(1H-1,3-benzodiazol-2-yl)-1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-(2-methylpropyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
(3S,4R)-4-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxylic acid
N-[2-(tert-butylsulfanyl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}propan-1-one
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
2,N4-dimethyl-N4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidine-4,6-diamine
3-[1-(oxan-4-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-[(4-methylphenyl)methyl]benzoyl}-2-(trifluoromethyl)morpholine
5-(methoxymethyl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)furan-2-carboxamide
N-[(3R,4S)-4-(propan-2-yl)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
methyl 2-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
[2-(5-propylpyrimidin-2-yl)phenyl]methanol
5-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-amino-4-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]pyrimidin-2-amine
3-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-ethyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-ethyl-5-[(3-methoxy-3-oxopropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
7-(prop-2-en-1-yloxy)-4-[2-(propylamino)pyrimidin-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(1,3-benzoxazol-2-yl)ethyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
1-(furan-2-ylmethyl)-4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]piperidine
6-ethyl-N-[3-(methylsulfanyl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-(1-acetylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide