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2-acetyl-8-(4-ethyl-5-methylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
3-(3-methoxypropyl)-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
5-{[5-(3-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-1,2,4-triazole
N-[(2-ethoxypyridin-3-yl)methyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]propanamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-2-yl}ethan-1-ol
2-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(1R,2S)-2-phenylcyclopropyl]acetamide
(1S,5R)-3-benzoyl-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
3-[1-(3,4-dimethyl-5-sulfamoylphenyl)-N-methylformamido]-N-methylbutanamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(pyridin-4-yl)ethyl]pyrrolidin-2-one
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]methyl}-2-chlorobenzamide
N'-(2-ethoxyphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]propanediamide
1-[1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)pyrrolidin-3-yl]-4-methylpiperazine
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
N-[3-(2-methylpyrimidin-4-yl)phenyl]-6-oxopiperazine-2-carboxamide
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
3-({[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)pyridin-2-amine
4-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide
1-(2-methoxy-4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-(4-fluoro-3-methoxyphenyl)-3-propylmorpholine-4-carboxamide
7-(cyclobutylmethyl)-2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
N,N-diethyl-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
4-{[(3-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 4-[3-(3-methylpiperidin-1-yl)propanoyl]piperazine-1-carboxylate
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(propan-2-yl)piperidine-3-carboxamide
7,7-dimethyl-2-{[1-(2-methylpropyl)piperidin-2-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(thiolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(4-methyl-1,3-thiazol-5-yl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)propanamide
N-(3-cyclopentylpropyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,4,6-trimethylpyrimidin-2-amine
1-ethyl-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(1R,6S)-9-methyl-3-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
(2R)-2-amino-3-methyl-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
N,6-dimethyl-4-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-dihydropyridine-3-carboxamide
1-{1-[(3-chloro-4,5-dimethoxyphenyl)methyl]azetidin-3-yl}piperidine
11-(1H-imidazol-4-ylmethyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
5-(3,3-diphenylpiperidine-1-carbonyl)-N,4-dimethyl-1,3-thiazol-2-amine
6-methyl-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(4aS,7aR)-1-(3-aminopropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(oxolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-cyclopentanecarbonyl-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S,4S,5R)-5-(2,3-difluorophenyl)-4-[(3-hydroxy-2,2-dimethylpropyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid