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1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-(3-fluorophenyl)piperidin-3-amine
(2R,6S)-2,6-dimethyl-4-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}morpholine
2-(4-fluorophenyl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
1-ethyl-3-(pyridin-2-ylmethyl)-8-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
5-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylpyrimidin-2-amine
3-methoxy-2-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]propanoic acid
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(6-methylpyridin-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-(3-hydroxypropyl)-N-[(2-methoxyphenyl)methyl]-3-methyl-1H-indole-2-carboxamide
2-(dimethylamino)-N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(3-methylphenyl)acetamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methylurea
N4-[(4-methoxypyridin-2-yl)methyl]-5-methylpyrimidine-2,4-diamine
1-(2-chloro-4-fluorophenyl)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)urea
(4-{[1-(1-benzyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[4-({[1-(1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
N-{2-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-oxoethyl}-N-(4-methylphenyl)methanesulfonamide
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)(oxan-4-ylmethyl)amine
3-(8-methylquinolin-5-yl)-1-(oxan-4-ylmethyl)urea
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1-(prop-2-en-1-yl)pyrrolidin-2-one
2-amino-N-{[1-(2-phenylethyl)pyrrolidin-3-yl]methyl}pyridine-4-carboxamide
8-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
7-methyl-3-(4-methylpyridine-3-carbonyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N2,N2,6-trimethylpyrimidine-2,4-diamine
N-cycloheptyl-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-[(4-phenyl-1,3-thiazol-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
5-ethyl-N,2,3-trimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(ethanesulfonyl)-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine
ethyl 2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-1,3-oxazole-4-carboxylate
3-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
N-methyl-5-{[methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})amino]methyl}pyrimidin-2-amine
8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dimethylquinoxaline-6-carbonyl)azetidine-2-carboxylic acid
1-[2-(4-hydroxypiperidin-1-yl)ethyl]-5,5-diphenylpiperidin-2-one
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
1-{4-oxo-4-[3-(2-phenylethyl)piperidin-1-yl]butyl}pyrrolidin-2-one
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(1,1-dioxo-1λ6-thiolan-3-yl)acetamide
dimethyl({3-[5-(1-methyl-1H-indol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl})amine
3-(2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-cyclopentanecarbonyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
methyl (2S,3S)-2-({[1-(2-carbamoylethyl)-1H-indol-3-yl]methyl}amino)-3-methylpentanoate
1-(2-fluoro-5-methanesulfonamidophenyl)-3-[1-(1-methyl-1H-imidazol-2-yl)butyl]urea
[1-({[1-(2-fluorophenyl)propan-2-yl]amino}methyl)cyclopentyl]methanol
N-(2-chloro-5-methylphenyl)-3-[(3-hydroxypiperidin-1-yl)methyl]benzamide
5-methanesulfonyl-2-methyl-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyrimidine
4-{[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}butan-1-ol