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5,6-dimethyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidine
ethyl 1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-3-carboxylate
1-benzyl-N,N-dimethyl-5-{[2-(methylsulfanyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
ethyl 3-[(2-methylphenyl)methyl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine-3-carboxylate
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-cyclohexyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
15-methyl-12-(4-methylpiperidine-1-carbonyl)-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(3-ethylphenyl)-4-(4-methoxyphenyl)-3-oxopiperazine-1-carboxamide
(2S,4S)-4-amino-1-(3-acetamidobenzoyl)-N-ethylpyrrolidine-2-carboxamide
1-(4-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}thiophen-2-yl)ethan-1-one
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]pyridazine
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2,8-diazaspiro[4.5]decane
1-(4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[(4-fluorophenyl)methyl]-5-[2-(pyrrolidin-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[3-(4-methoxyphenyl)propyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[2-(methylsulfanyl)ethyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
4-(4-methylpyridin-3-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,8aR)-1-(4-hydroxybutyl)-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
(3S,4S)-4-cyclopropyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidine-3-carboxylic acid
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-[2-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
N6-(3-methoxypropyl)-N5-methyl-N5-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-(5-fluoro-2-methoxyphenyl)-4-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
6-methyl-4-[2-oxo-2-(1,3-thiazolidin-3-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-amino-4-cyclopropyl-6-(3-methoxyphenyl)pyridine-3-carbonitrile
3-[3-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-4-yl]pyridine
4-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-N,N-dimethylpiperazine-1-carboxamide
1-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
benzyl(methyl){[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-oxazol-5-yl]methyl}amine
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-triazole-5-carboxamide
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
2-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}morpholin-2-yl)ethan-1-amine
2-chloro-6-methoxy-4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenol
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-(pyrimidin-2-yl)-1,4-diazepane
methyl 2-[(3-methylbutyl)sulfamoyl]-6-(quinolin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]pyridine-3-carbonitrile
5-{[benzyl(methyl)amino]methyl}-N-[(1-ethylcyclobutyl)methyl]-1,2-oxazole-3-carboxamide
dimethyl({4-[1-(pyridin-4-ylmethyl)piperidin-2-yl]phenyl}methyl)amine
ethyl 1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxylate
(4aR,7aS)-1-[2-(4-methylpiperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine