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N-[(1,2-dimethyl-1H-indol-3-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[5-(2,6-dimethylphenyl)-1H-indazol-1-yl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3aS,6aS)-5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-cyclohexyl-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
1-cyclopropyl-5-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
4-fluoro-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-(6-methoxypyrimidin-4-yl)-3-(2-methylphenyl)pyrrolidin-3-ol
3-(tert-butylsulfamoyl)-N-[(1-methylpiperidin-3-yl)methyl]-5-[(2-methylpropyl)amino]benzamide
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
3-(5-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
6-{[(1R,5S,6R)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-[(4-hydroxyphenyl)methyl]-1-(2-methylpropyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
6-[1-(carbamoylmethyl)piperidine-4-carbonyl]-N,1-dimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[2-(pyridin-2-ylsulfanyl)acetyl]-decahydro-2,7-naphthyridine-2-carboxamide
4-(2,1,3-benzoxadiazol-4-yl)-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N,N-dimethyl-2-{[3-(2-oxoazepan-1-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[(2S,4S)-4-fluoro-1-[4-(thiophen-2-yl)butanoyl]pyrrolidin-2-yl]methyl}-3-methylbutanamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}acetamide
4-benzyl-1-[(2-methoxypyridin-3-yl)methyl]pyrrolidin-2-one
4-(2-methyl-6-{1-[(2S)-pyrrolidine-2-carbonyl]piperidin-4-yl}pyrimidin-4-yl)morpholine
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
methyl N-{1-oxo-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-2-yl}carbamate
N-methyl-2-(morpholin-4-yl)-N-(prop-2-en-1-yl)benzamide
[(3R,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(hydroxymethyl)-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}azepan-4-ol
5-(2-phenyl-1H-imidazol-1-yl)pyridine-3-carboxamide
N-benzyl-N-ethyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-methyl-N-(pyrazin-2-ylmethyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
(3S)-N,N-dimethyl-1-{[(1s,4s)-4-aminocyclohexyl]methyl}azepan-3-amine
3-[(1-benzothiophen-5-ylmethyl)amino]-N-(2-fluorophenyl)propanamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
3,3-dimethyl-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-ethyl-1,3,4-oxadiazol-2-amine
2-{4-[4-(1H-imidazol-1-yl)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
[1-(4-aminopyrimidin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-({1-[(3-fluorophenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
3-propyl-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-3-carboxylic acid
N-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
9-(8-chloroquinoline-2-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
2-(4-{[(4-cyano-2-fluorophenyl)carbamoyl]amino}piperidin-1-yl)-N-cyclopropylacetamide
N-cyclopentyl-2,5-dimethyl-N-(prop-2-en-1-yl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(1-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl)dimethylamine
2-[(1S,5R)-3-(2,1,3-benzoxadiazol-4-ylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-amino-3-ethyl-N-[(2-methylphenyl)methyl]-N-(2-methylpropyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
9-[2-(2-hydroxyethoxy)ethyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine