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1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-4-(4-methoxyphenyl)butan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-imidazol-2-yl}pyridine
benzyl N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
3-(2H-1,3-benzodioxol-5-yl)-5-[4-(methylsulfanyl)butan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-methyl-N-(pyridin-3-ylmethyl)-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5,5-dimethyl-3-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]-1,3-oxazolidine-2,4-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-3-ol
methyl 4-{[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]methyl}benzoate
5-{[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-{4-[(3-hydroxyphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
1-{[1-(2-fluorophenyl)cyclopentyl]methyl}-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
2-[1-(furan-3-ylmethyl)-4-(1H-1,2,3-triazole-5-carbonyl)piperazin-2-yl]ethan-1-ol
4-chloro-N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
1-(3-chloro-4-methylphenyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-amine
9-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(1-cyclohexylpiperidin-3-yl)methyl][(1-phenyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-4-methylpiperidine-1-sulfonamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(5-phenylfuran-2-yl)methyl]acetamide
1-{4-[({[2-(dimethylamino)pyridin-3-yl]methyl}amino)methyl]thiophen-2-yl}ethan-1-one
N-ethyl-3,5-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-indole-2-carboxamide
3-butyl-4-[2-(1H-imidazol-2-yl)benzoyl]-1-methylpiperazin-2-one
N-(1-propyl-1H-pyrazol-5-yl)-2-(4-{thieno[3,2-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
5-fluoro-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-2,3-dihydro-1H-indol-2-one
5-fluoro-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-indole-2-carboxamide
2,4-dichloro-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenol
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-{5-[(2,2-dimethylmorpholin-4-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
6-(4-{[1-(6-methylpyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)-2-(propan-2-yl)pyrimidin-4-ol
6-[(3-fluorophenyl)methoxy]-4-(4-methyl-1H-imidazole-2-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
1-({1-[6-(2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-methyl-3-(piperidine-1-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
[(2,3-dimethoxyphenyl)methyl]({[2-(2-methoxyphenyl)-6-methylquinolin-3-yl]methyl})amine
3-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
6-[(diethylamino)methyl]-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(4S)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-[(4-phenyloxan-4-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-methyl-7-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2,4-dichlorophenoxy)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
(2-{[(2-methoxypyrimidin-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
4-(cyclopropylmethyl)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
1-(2-methylphenyl)-4-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperazin-2-one
6-[1-(1-benzoxepine-4-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
3-hydroxy-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
5-acetyl-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide