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N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1-methylpiperidine-4-carbonyl)piperidine
N-(1-{1-[(3,4-dimethoxypyridin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
5-methyl-3-(1,3-thiazol-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(pyridine-3-carbonyl)piperazine
(3R,4S)-1-(2-ethoxyethyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
3-methyl-1-[4-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}sulfonyl)phenyl]urea
3-[methyl({5-methylpyrazolo[1,5-a]pyrimidin-7-yl})amino]propanamide
2-chloro-4-acetamido-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]benzamide
N-(2-hydroxyethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(1-phenoxypropan-2-yl)({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[(3-methylquinoxalin-2-yl)methyl]cyclopropanamine
6-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-methyl-4-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-({[(5-ethylfuran-2-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
N-{1-[1-(5-acetylthiophene-2-carbonyl)piperidin-4-yl]-2-(4-fluorophenyl)ethyl}-N-methyl-3-(methylsulfanyl)propanamide
1-(carbamoylmethyl)-N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]morpholin-2-yl}methanamine
[(2S)-1-[(1,3-diphenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl]methanol
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-4,4,4-trifluorobutan-1-one
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3-(1H-indol-2-ylmethyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-(3,4-dimethoxyphenyl)-1-(oxan-2-ylmethyl)-1H-imidazole
2-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
6-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
4-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
4-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]thiomorpholine
1-{4-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-ylmethyl]phenyl}-1H-imidazole
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
3-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-[5-(5-methyl-1,3-oxazol-4-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{[(3S,4S)-3-hydroxy-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl]methyl}-2,5-dimethylfuran-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
2-(2-{[(4aS,7aR)-4-acetyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}phenoxy)acetic acid
N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
2-{1-cyclopentyl-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(3aR,7aS)-2-[(4-methanesulfonylphenyl)methyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-methoxypyrimidine
N-[(3-methoxyphenyl)methyl]-3-{1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-3-yl}propanamide
(2S,4R)-1-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-4-amino-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(pent-2-yn-1-yl)piperidine
N-[(1S)-1-(3-methoxyphenyl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2,5-dimethyl-4-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-oxazole
methyl 2-(cyclopropylsulfamoyl)-6-(4-phenylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate