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4-(2-chloro-4-fluorophenyl)-5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[(3-methoxyphenyl)methyl]-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-cyclopentyl-4-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetyl]piperazin-2-one
methyl 5-[4-(propan-2-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-(1-methyl-1H-indazol-5-yl)-3-[(2-methylphenyl)methoxy]azetidine-1-carboxamide
N-(2-fluorophenyl)-3-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-(3-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-3-oxopropyl)-4-fluorobenzamide
1,2-dimethyl-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
1-[(3-methoxyphenyl)methyl]-4-(1-methylazepane-2-carbonyl)piperazin-2-one
(3aR,6aR)-2-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-5-(3-methylbut-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4S)-1-cyclohexyl-N-ethyl-4-[2-(3-fluorophenyl)acetamido]pyrrolidine-2-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2-methanesulfonylethyl)acetamide
N-(5-methyl-1,2-oxazol-3-yl)-2-[(2S)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
(2S,3R)-3-hydroxy-2-[4-(2-phenylphenyl)-1H-1,2,3-triazol-1-yl]butanoic acid
2,3-dimethyl-6-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-cyclohexyl-4-(1H-pyrazol-3-yl)-N-(pyridin-2-ylmethyl)benzamide
6-(2,5-dimethylfuran-3-yl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[(3-methylthiophen-2-yl)methyl]-N-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]cyclopropanamine
1-(4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}benzoyl)pyrrolidine
N-(2-chloro-5-methylphenyl)-4-(3-hydroxypiperidin-1-yl)piperidine-1-carboxamide
N3-ethyl-N5-[1-(furan-2-yl)ethyl]-N3-(2-methylprop-2-en-1-yl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopentyl-4-[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]benzonitrile
6-[(3-fluorophenyl)methyl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
ethyl 3-benzyl-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine-3-carboxylate
1-[(3-chloro-4-fluorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1,3-thiazol-2-yl)piperidine-4-carboxamide
7-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-phenyl-5-(4,4,4-trifluorobutyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
7-methoxy-3-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1-propylpiperidin-4-amine
4-(1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyridine
2-methoxy-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyridine
6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carbonitrile
3-(2-ethoxypyridin-3-yl)-5-(morpholine-4-sulfonyl)benzoic acid
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-phenylmethanesulfonamide
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
5-ethyl-1'-[3-(1H-imidazol-2-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-fluoro-N,N-dimethyl-2-(1-phenyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
N,1-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-indole-6-carboxamide
1-(1'-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-propoxypiperidine-1-carboxamide
(1S,5R)-6-(3,4-difluorobenzenesulfonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-hydroxybenzamide
1-[3-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1-methylpiperidin-4-yl)piperazine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide