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5-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
ethyl({imidazo[1,2-a]pyrimidin-6-ylmethyl}){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-4-ol
(9aR)-8-(cyclopropylmethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-amino-N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)cyclopentane-1-carboxamide
N-[2-(4-propoxyphenyl)ethyl]morpholine-2-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-2-amine
1-(2-methylphenyl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1,4-diazepane
2-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-methyl-6-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)pyridine
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
1-ethyl-4-{[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
(1R,9S)-5-amino-12-methyl-3-[3-(1H-pyrazol-1-yl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-[5-methyl-4-(5-methylthiophene-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
[4-({2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-4-yl}methyl)-1,4-oxazepan-6-yl]methanol
3-(2-methylquinolin-5-yl)phenol
({1-[2-(2-ethylmorpholin-4-yl)ethyl]-3-methyl-1H-pyrazol-4-yl}methyl)[(2-methylphenyl)methyl]amine
3-{3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}pyridine
2-methoxy-5-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
1-(5-methyl-1-benzofuran-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-{1-[1-(4-ethenylbenzoyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
N-methyl-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-[2-({6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidin-3-yl}formamido)ethyl]acetamide
3-hexyl-8-(4-methyl-1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-({4-[4-(cyclopentylcarbamoyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}sulfonyl)thiophene-2-carboxylate
1-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3,3-bis(propan-2-yl)urea
2-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N-methylpyridine-4-carboxamide
3-(6-cyanopyridin-3-yl)-1-(3-methoxypropyl)-1-[(4-methylphenyl)methyl]urea
3-methanesulfonyl-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(2-amino-6-methylpyrimidin-4-yl)-1-[(4-fluorophenyl)methyl]piperazin-2-one
4-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
(3R,5S)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
6-[2-(piperidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
4-(methoxymethyl)-3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-5-methyl-1,2-oxazole
3-(2-ethylbutyl)-8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(methoxymethyl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylthiophene-2-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
ethyl(methyl){1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}amine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-phenylethyl)acetamide
4-{1-[2-(phenylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl}benzoic acid
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
2-methoxy-1-[1'-(6-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]piperidine-1,3-dicarboxamide
1-(2-aminoethyl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(methoxymethyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrrolidine
3,5-dimethyl-1-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidin-3-yl)-1H-pyrazole
3-[3-({[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}methyl)-1H-indol-1-yl]propanamide
1-(1,4-dithiepan-6-yl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
(3S,4R)-1-(oxane-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid