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1-cyclopentyl-4-({methyl[(4-oxo-4H-chromen-3-yl)methyl]amino}methyl)pyrrolidin-2-one
2-amino-4-(3-methylthiophen-2-yl)-6-(oxolane-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-methyl-2-(phenylamino)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
ethyl 1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(3-cyclobutyl-1H-1,2,4-triazol-5-yl)-1-methyl-1H-indole
methyl({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(pyridin-2-ylmethyl)amine
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-N-(2,4-dimethoxyphenyl)propanamide
3-ethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1,2-oxazole-5-carboxamide
1-methyl-4-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperazine
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}cyclohexanamine
N-[(2-phenoxypyridin-3-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(3aR,5S,6S,7aS)-2-[(6-methoxy-2H-chromen-3-yl)methyl]-octahydro-1H-isoindole-5,6-diol
(3S,4R)-3-benzyl-4-methyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-ol
2-phenyl-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-benzyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(piperidin-1-yl)ethyl]amino}methyl)piperidin-2-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
4-(2H-1,3-benzodioxole-5-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 1-[1-benzyl-5-(ethylcarbamoyl)-4-oxo-1,4-dihydropyridine-3-carbonyl]piperidine-2-carboxylate
1-[1'-(2,5-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-[4-(dimethylamino)azepane-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
(2E)-1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}-3-phenylprop-2-en-1-one
3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-7-(2-methoxyacetamido)-N,1-dimethyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
(1R,6S)-9-methyl-3-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
N-methyl-2-propyl-N-[1-(1,3-thiazol-2-yl)ethyl]pyridine-4-carboxamide
3-phenoxy-N-{1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(thiophen-3-yl)propanamide
benzyl(benzylsulfamoyl)(3-hydroxy-2-methylpropyl)amine
(3S,4R)-1-(3-methyloxetane-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
3-(oxolan-3-yl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-[(3R,4S)-1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]ethane-1-sulfonamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-ethyl-1H-pyrazole-4-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
4-(2,5-dimethylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-(5-acetamido-2-methoxyphenyl)-3-phenylpiperazine-1-carboxamide
5-(furan-2-ylmethyl)-5-[3-oxo-3-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propyl]pyrrolidin-2-one
2-[2-(dimethylamino)ethyl]-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)methyl]-6-methylquinolin-4-ol
4-[({1,9-dioxaspiro[5.5]undecan-4-yl}amino)methyl]benzene-1-sulfonamide
N-cyclohexyl-1-ethyl-3-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
4-methyl-9-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
ethyl 4-benzyl-1-(4-acetamidobenzenesulfonyl)piperidine-4-carboxylate
1-benzyl-8-(butan-2-yl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-4-carboxamide
N-ethyl-N-(2-hydroxy-3-phenoxypropyl)-3-(4-hydroxyphenyl)benzamide