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4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
5,6-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyridine-3-carboxamide
6-(aminomethyl)-2-(4-{[methyl(2-phenoxyethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(thiomorpholine-4-sulfonyl)-5-(1H-1,2,3-triazol-1-yl)benzoic acid
1-[1-(hydroxymethyl)cyclopropanecarbonyl]-4-(5-methyl-1,3,4-thiadiazol-2-yl)-1,4-diazepane-6-carboxylic acid
2-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2R)-2-phenyl-2-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)ethan-1-ol
N-(3,4-dimethylphenyl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
2-chloro-N-({1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}methyl)benzamide
3-{[2-(dimethylamino)-2-(3-methylphenyl)acetamido]methyl}-1,2,4-oxadiazole-5-carboxamide
3-hydroxy-3-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]-1-(2-phenylethyl)piperidin-2-one
1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-({5-[(3-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-{3-[({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}ethan-1-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(propan-2-yl)pyrimidine-4-carboxamide
(1R,3S)-3-[4-(3-chloro-4-fluorophenyl)piperazine-1-carbonyl]cyclopentane-1-carboxylic acid
2-amino-4-(2-butyl-1H-imidazol-4-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-(pyridin-2-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
[3-(cyclopropylmethyl)-1-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-3-yl]methanol
2-{imidazo[1,2-a]pyridin-3-yl}-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
methyl 2-(cyclohexylsulfamoyl)-6-(4-methylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[5-(ethanesulfonyl)thiophen-2-yl]quinoline
3-(pyridin-4-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(3S,7S,8aS)-7-{[(2,5-difluorophenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[1-(pyridazine-4-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-(3-methoxyphenyl)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
5-[({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,5-difluoro-4-methoxybenzamide
methyl 4-[({1-[4-(2,4-dimethylbenzamido)phenyl]piperidin-4-yl}amino)methyl]benzoate
3-[(oxolan-3-yl)sulfamoyl]-N-[2-(piperidin-1-yl)ethyl]benzamide
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(furan-2-carbonyl)piperidine
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-2-[3-(pyridin-3-ylmethyl)piperidin-1-yl]pyrimidine
4-[(3-acetamidopyrrolidin-1-yl)methyl]-N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)benzamide
1-cyclohexyl-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-(pyridin-2-ylmethyl)urea
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopentyl-3-[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
2-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
1-methyl-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-3-carbonyl]-N,N-dimethylpyrrolidin-3-amine
(5S)-5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)butan-1-one
1-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]-3-phenylpropan-1-ol