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N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)acetamide
2-[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
8-[2-(1H-imidazol-2-yl)benzoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-phenylcyclohexane-1-carboxamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
1-(cyclopent-1-ene-1-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
4-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4-(pyridin-4-yl)pyrimidin-2-amine
2-{1-[(4-ethoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
(3aR,6aS)-2-methyl-5-[(6-methylquinolin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
3-(2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(4-phenoxybenzoyl)piperidine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(hydroxymethyl)benzamide
8-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aR,6aS)-5-[1-(2-methoxyphenyl)piperidin-4-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
5-ethyl-N-[3-(oxolan-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidin-3-amine
1-[(2,3-difluorophenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-cyclopropyl-1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
2-(1H-imidazol-1-yl)-1-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
1-[(3,5-dichloro-2-methoxyphenyl)methyl]piperidine-3-carbonitrile
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}acetamide
2-methoxy-5-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-({1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}methyl)-4-phenylbenzamide
4-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-N,N-dimethylbenzamide
N-{[3-(carbamoylmethyl)-1-[4-(propan-2-yl)phenyl]-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
N-[3-(4-hydroxyphenyl)propyl]-2-(1H-imidazol-2-yl)benzamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-propyl-1H-pyrazole-5-carboxamide
6-[3-(1-methoxyethyl)phenyl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-[(1R,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-[(4-methylphenyl)methyl]propanamide
2-(1H-1,3-benzodiazol-1-yl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
2-(dimethylamino)-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
(1R,5S,6S)-N-cyclopentyl-3-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-[2-(5-methylthiophen-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(2-fluorophenoxymethyl)-3-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
5-methyl-3-[3-(1H-pyrazol-1-yl)propyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(4-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
8-[3-(pyridin-3-yl)propyl]-8-azaspiro[4.5]decane-7,9-dione
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide