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ethyl 2-[1-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)piperidin-2-yl]acetate
6-methyl-1-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1,2-dihydropyridin-2-one
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxypyridine
1-methyl-3-{[1-(6-methylpyridazin-3-yl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({1-[2-(1H-pyrazol-1-yl)butanoyl]piperidin-4-yl}methyl)benzoic acid
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-3-carboxamide
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-(methoxymethyl)-1H-1,2,4-triazole
2-[4-(5-methyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-N-(pyridin-3-yl)acetamide
4-(3,3-diphenylpiperidin-1-yl)-N,N-dimethyl-4-oxobutanamide
4-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]-1,4-oxazepan-6-ol
1-(2,3-dihydro-1H-isoindol-2-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-({4-hydroxy-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]azepan-4-yl}methyl)-2-phenylacetamide
3,5-dichloro-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-methylbenzamide
(2R)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]-3-(3,4,5-trifluorophenyl)propanoic acid
N,N-dimethyl-4-[4-({[1-(morpholin-4-yl)cycloheptyl]methyl}amino)piperidin-1-yl]benzamide
(2S,4R)-4-amino-1-(4-methoxycyclohexanecarbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[3-(diethylamino)pyrrolidine-1-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
2,6-dimethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}pyridine-4-carboxamide
2-(4-{5-amino-4-cyano-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-trien-3-yl}-2-methoxyphenoxy)acetamide
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-chloro-N,N-bis(2-hydroxyethyl)naphthalene-1-carboxamide
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2E)-1-[(4aR,8aS)-6-(2-methoxyacetyl)-decahydro-1,6-naphthyridin-1-yl]-3-(2-chlorophenyl)prop-2-en-1-one
2-[(3-methylbut-2-en-1-yl)(thiophen-3-ylmethyl)amino]butan-1-ol
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-4-ol
N-cyclopropyl-2-[3-(3-ethylphenoxy)azetidin-1-yl]pyridine-4-carboxamide
(3-ethyl-1-{3-[(thiophen-2-ylmethyl)amino]benzoyl}piperidin-3-yl)methanol
4-(4-methoxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-oxobutanamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(1H-imidazol-2-yl)benzamide
1-[1-(6-aminopyridine-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
1-(4-fluorophenyl)-4-(pyrazine-2-carbonyl)-1,4-diazepane
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-(3-methoxyphenyl)piperazin-2-one
4-(hydroxymethyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]azepan-4-ol
2-methoxy-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-5-sulfamoylbenzamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-ethoxypropan-1-one
1-[3-(5-methylfuran-2-yl)benzoyl]-4-(thian-4-yl)piperazine
1-(3-methoxyphenyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-2-one
N-[(1R,2R)-2-(benzyloxy)cyclohexyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
4-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-N-(1,3-thiazol-2-yl)benzamide
3-[(dimethylamino)methyl]-1-(2,2-diphenylethyl)piperidin-3-ol
N-(2,5-dimethoxyphenyl)-2-[2-(pyrrolidin-1-ylmethyl)-4-(thiophen-2-yl)phenoxy]acetamide
7-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N,1,7-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-indole-2-carboxamide