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N-(3-phenylprop-2-yn-1-yl)-N-propyl-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetamide
(4aS,8aR)-N-[2-(2-fluorophenyl)ethyl]-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3,3,4,4-tetrafluorobutyl)pyrrolidine-3-carboxylic acid
1-(4-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
methyl 6-oxo-4-[(1E)-1-phenylprop-1-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
7-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
2,4,6-trimethyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}benzamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1-methyl-5-oxopyrrolidine-3-carboxamide
2-{[(2E)-3-phenylprop-2-en-1-yl]({[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl})amino}ethan-1-ol
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
4-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-1-methyl-1H-pyrazole
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(2-methoxyquinolin-3-yl)-N-methylpyridine-3-carboxamide
6-methoxy-N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 4-(4-{[2-(methoxymethyl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
4-(3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propoxy)benzamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
[1-(ethylsulfanyl)propan-2-yl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-{4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
3-(3,4-dimethyl-1H-pyrazol-5-yl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)propan-1-one
1-{3-[({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]propyl}pyrrolidin-2-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-azaspiro[5.5]undecan-9-amine
4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}-2,3-dihydro-1H-inden-1-one
2-(3,4-dichlorophenyl)-4-[(2-ethylpyrimidin-5-yl)methyl]morpholine
6-methoxy-2-oxo-N-[3-(phenylsulfanyl)propyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[1-(1H-1,3-benzodiazole-5-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
8-(2,5-dimethylbenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N3-benzyl-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
methyl 3-{[5-(hydroxymethyl)furan-2-yl]methyl}-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,3R)-N1-[2-(benzyloxy)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(4-cyano-2-fluorophenyl)-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclobutanecarboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(2-hydroxy-3-methylbenzoyl)pyrrolidine-2-carboxamide
5-acetyl-6-methyl-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
12-[4-(dimethylamino)azepane-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
[1-(isoquinolin-1-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
4-{[3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]methyl}morpholine
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-methyl-5-[(methylsulfanyl)methyl]-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-(2-methoxyethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
diethyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})amine
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
N-cyclohexyl-2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}butanamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-hydroxy-4-(methylsulfanyl)butan-1-one
3-{2-[2-(propan-2-yloxy)phenoxy]ethyl}-1,3-diazinane-2,4-dione
3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methyl-2,8-diazaspiro[4.5]decane
3-({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione