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2-(2,4-difluoro-3-methoxybenzoyl)-2,7-diazaspiro[4.5]decane
4-[4-(3-fluorobenzoyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-chloro-9-(2-methoxyphenyl)-15-methyl-N-(2-methylpropyl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)pyrrolidine-3-carboxylic acid
N5-(2,3-dihydro-1H-inden-2-yl)-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethyl-4-oxobutanamide
1-{3-[3-(benzyloxy)azetidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
8-methoxy-2-methyl-5-[2-(piperazin-1-yl)phenyl]quinoline
3-cyclohexyl-1-[2-(ethylsulfanyl)ethyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-(4-{[6-methoxy-3-oxo-4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}phenyl)acetamide
N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(1-methyl-1H-pyrazole-5-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
2-{5-[6-amino-5-cyano-4-(trimethyl-1H-pyrazol-4-yl)pyridin-2-yl]thiophen-3-yl}acetic acid
N-(pyridin-4-ylmethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide
2-[5-(3-methyl-5,6,7,8-tetrahydroisoquinolin-4-yl)-2H-1,2,3,4-tetrazol-2-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
1-{2-[4-(pyridin-3-yloxy)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
3-methyl-2-phenyl-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
5-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(2-methylpropyl)-1H-imidazole
2-{[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
1-{2-[1-(3,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)-2-phenylethan-1-ol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-(2-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-2-yl}ethyl)phenol
3-(oxolan-3-yl)-5-(3-phenylphenyl)-1,2,4-oxadiazole
5-(3-benzoylpiperidine-1-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
4-(2,4-difluoro-3-methoxybenzoyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-{[(2,6-dimethoxypyrimidin-4-yl)amino]methyl}-3,4-dihydroquinazolin-4-one
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
1-({1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)pyrrolidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(dimethyl-1,2-oxazol-4-yl)propanamide
7-cyclohexyl-2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-(quinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
[(2-methoxy-5-{[3-(2-methoxyethyl)piperidin-1-yl]methyl}phenyl)methyl]dimethylamine
2,3,5-trimethyl-N-[1-(3-methylpyridin-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazinane
4-ethyl-3-{1-[2-(1H-indazol-3-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methyl-2-({4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}methyl)-5,6,7,8-tetrahydroquinazoline
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
(3S,9aR)-3-(hydroxymethyl)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2,6,8-trimethyl-4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]quinoline
N-(3,5-dimethylphenyl)-6-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{2-[2-(5-fluoro-2-methoxyphenyl)phenoxy]ethyl}-1H-imidazole
N-[2-(1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]acetamide