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1-{5-cyclopentyl-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
6-(3-methyl-3-phenylpiperidin-1-yl)pyrimidin-4-amine
N-{4-[2-(dimethylamino)ethoxy]-1-(4-fluorophenyl)-1H-indazol-3-yl}oxolane-2-carboxamide
5-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-phenylpyrimidin-4-ol
N-methyl-2-[methyl({5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl})amino]acetamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
N,N-dimethyl-5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[2-(morpholin-4-yl)quinolin-3-yl]methyl}amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(2-methyl-1,4-oxazepan-4-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]acetamide
2-{1-[(3-methoxyphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}thieno[3,2-d]pyrimidin-4-amine
3-(2H-1,3-benzodioxol-5-yl)-N-[3-(1H-imidazol-1-yl)propyl]-3-phenylpropanamide
3-{5-[(3-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2-hydroxyethyl)propanamide
5-(1,3-thiazolidine-3-carbonyl)-1,3-benzothiazol-2-amine
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)urea
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{[2-({[1-(methoxymethyl)cyclopropyl]methyl}carbamoyl)phenyl]amino}acetic acid
3-[2-(4-methanesulfonylphenyl)-4-methylphenyl]-1,3-oxazolidin-2-one
6-{3-[(5-methylpyridin-2-yl)amino]propyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
7-(1,3-benzothiazol-2-yl)-4-(morpholine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S)-1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
3-[1-(5-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]propanoic acid
(2R,3R,6R)-3-phenyl-5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2,4-dimethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)pyrimidine-5-carboxamide
N-(1-acetylpiperidin-3-yl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(benzylsulfamoyl)[3-(4-methoxyphenyl)propyl]amine
(2R,6S)-4-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[(1S,5R)-6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-[4-(2-ethylbutyl)piperazin-1-yl]-2-[2-(3-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[2-methoxy-4-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-cyclopropyl-6-oxo-N-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
3-chloro-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-N-(oxolan-2-ylmethyl)acetamide
1-methyl-3-[1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]piperidine
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-cyclobutyl-7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
1-ethyl-3,5-dimethyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
2-(methylsulfanyl)-5-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}pyrimidine
4-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
3-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-N-(2,5-dimethoxyphenyl)-3-oxopropanamide
3-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(4S)-3-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-4-phenyl-1,3-oxazolidin-2-one
7-acetamido-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-acetyl-8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid