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6-(1,4-diazepan-1-ylmethyl)-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-(3,4-difluorophenyl)piperidin-3-amine
N-methyl-2-[methyl(pyridin-2-ylmethyl)amino]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-{4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]-6-methylpyrimidin-2-yl}phenol
2-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
(2H-1,3-benzodioxol-4-ylmethyl)(ethyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amine
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}butanamide
3-({1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
3-({2-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
6-(3-ethylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
methyl 2-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}piperidine-1-carboxylate
N-[(3S,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
7-(6-chloropyridazin-3-yl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(3-chloro-4-methoxyphenyl)methyl]-2-(methoxymethyl)piperidine
(2S,4R)-4-[4-({[(3-chloro-4-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
8-(1-benzofuran-2-ylmethyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-[(3-chloro-4-fluorophenyl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[1-(2,2,6,6-tetramethylpiperidin-4-yl)piperidin-3-yl]oxy}methyl)pyridine
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-2-(2-methoxyethyl)piperidine
2-(oxan-2-ylmethoxy)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
(1S,5R)-6-(3,4-dimethylbenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-chloro-5-methylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-3-amine
3-[(diethylamino)methyl]-N-(1H-indazol-6-yl)benzamide
N-(3-methoxyphenyl)-3-[(2-methylbutyl)amino]-5-(pyrrolidine-1-sulfonyl)benzamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-phenyl-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,3-oxazole
4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
1,4-dimethyl 2-{[1-(4-{[(2-fluorophenyl)methyl]carbamoyl}phenyl)piperidin-4-yl]amino}butanedioate
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2,5-dimethyl-3-{4-[(2-methylfuran-3-yl)methyl]piperazin-1-yl}pyrazine
1-{2-[ethyl(phenyl)carbamoyl]ethyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
2-hydroxy-4-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}quinoline-6-sulfonamide
2-(2-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}ethyl)pyridine
3-[(4aR,7aS)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-cyclohexyl-N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-1H-pyrazole-4-carboxamide
N'-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)ethanediamide
1-(azocan-1-yl)-3-(2-methoxy-5-{[(2-phenoxyethyl)amino]methyl}phenoxy)propan-2-ol
(3aS,6aS)-2-[(4-chlorophenyl)methanesulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
1-(oxolane-2-carbonyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
N-[2-(dimethylamino)ethyl]-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(3-{1-[2-(dimethylamino)ethyl]-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(trifluoromethyl)benzamide