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N3-(adamantan-1-ylmethyl)-N3-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]acetamide
1-{[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
8-(1-hydroxypropan-2-yl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(4-cyclopropyl-5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline
ethyl 1-(tert-butylcarbamoyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
7-{2-amino-6-[(4-methylphenyl)sulfanyl]pyrimidin-4-yl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[4-(2,4-dimethoxyphenyl)-6-ethylpyrimidin-2-yl]morpholine
(3S,5R)-1-(pyridin-2-ylmethyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-(naphthalen-2-ylmethyl)-1,3λ6,4-oxathiazinane-3,3-dione
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-methyl-3-phenylpiperidine
4-(1H-imidazol-1-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}butan-1-one
2-methoxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropane-1-carboxamide
2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-N-(thiophen-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3,5-dimethyl-2-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-indole
(3R,4S)-4-(3-methoxyphenyl)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-amine
4-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-(5-methyl-2-pentanamidophenyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-2-ylmethyl)piperazine
5-{3-[2-(2,6-dimethoxyphenyl)-1H-imidazol-1-yl]-4-methylphenyl}-1H-1,2,3,4-tetrazole
{2-[2-(furan-2-yl)-1H-imidazol-1-yl]-1-(3-methylphenyl)ethyl}dimethylamine
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(naphthalene-2-carbonyl)piperidine
2-(2,6-dichlorophenyl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-(2-chlorophenyl)-1-methylpyrrolidine-2,5-dione
N-(4-cyano-2-ethylphenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-{5-[2-(2-methylphenyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-ol
(1S,5R)-6-(cyclopropylmethyl)-3-[(3-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxy-6-methylphenyl)-3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carboxamide
(1S,3R)-3-amino-N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-2-ylmethyl)cyclopentane-1-carboxamide
(3S,4S)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidine-3-carboxylic acid
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-[methyl(phenyl)amino]ethan-1-one
1-methyl-3-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
9-(3-hydroxypyridine-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-N-(1-methylpiperidin-3-yl)pyrimidin-2-amine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)piperidin-3-ol
5-{4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-6-methoxypyrimidin-4-amine
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methoxypyridine-3-carbonitrile
3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-(pyrrolidin-1-yl)pyridazine
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]oxolane-2-carboxamide
(3S)-3-ethyl-4-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carbonyl}morpholine
({5-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(2-acetamidophenyl)-2-({[3-(trifluoromethoxy)phenyl]methyl}amino)acetamide
N-{2-[3-(dimethylamino)phenoxy]propyl}-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine