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1-[5-(4-methanesulfonylphenyl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
2-[methyl({4-methyl-5-[1-(3-methylbenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2-ethyl-N,4-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-oxazole-5-carboxamide
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-2-propyl-1,3-thiazole-4-carboxamide
N5-cyclopropyl-N6-[phenyl(pyridin-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(3-fluoro-4-methoxybenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-{[1-(4-cyclopentyl-1,4-diazepan-1-yl)-1-oxopropan-2-yl]sulfanyl}-6-methyl-3,4-dihydropyrimidin-4-one
1-(4-methoxyphenyl)-2,2-dimethyl-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
2-{4-[3-methyl-1-(pentan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}ethan-1-ol
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
1-methyl-N-[(3R,5S)-1-methyl-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-5-phenyl-1H-pyrrole-2-carboxamide
4-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
1-(2,3-dihydro-1H-inden-4-yl)-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
4,5-dimethyl-2-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole
8-methyl-2-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]-2,8-diazaspiro[4.5]decane
5-[2-(3-chloro-1H-1,2,4-triazol-5-yl)ethyl]-3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
N-[2-(1H-imidazol-1-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-cyclopentyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
(1S,5R)-6-(cyclopropylmethyl)-3-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(4-cyclopentylpiperazin-1-yl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
6-(methoxymethyl)-1-methyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-phenylpropyl)-4-(thiophene-3-carbonyl)-1,4-diazepane
3-[(2-methoxyethyl)(pyridin-4-ylmethyl)carbamoyl]benzoic acid
4,6-dimethyl-13-[(1s,4s)-4-aminocyclohexyl]-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
1-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-2-ol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}-4-[2-(pyridin-4-yl)ethyl]piperazine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
4-amino-2-(5-phenylthiophen-2-yl)pyrimidine-5-carbonitrile
1-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
6-methyl-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
3-[4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
6-chloro-N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(4-{1-[2-(1H-pyrrol-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)pyridine
6-fluoro-2-[2-(methoxymethyl)pyrimidin-5-yl]-4-(1,4-oxazepane-4-carbonyl)quinoline
6-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylfuran-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(hydroxymethyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-4-(1H-imidazol-1-yl)butan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methyl-2-[(propan-2-yl)amino]benzamide
(3aS,6aS)-2-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
1-cyclopentyl-N-(3-methyl-1,2-thiazol-5-yl)-6-oxopiperidine-3-carboxamide
1-[(2R)-2-hydroxy-2-phenylacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(2-methylpropyl)-8-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one