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N-propyl-2,8-diazaspiro[4.5]decane-2-carboxamide
(1S,5R)-3-[2-(benzyloxy)ethyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-methyl-6-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
7-(3-methoxyphenyl)-2-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3R,4R)-3-hydroxy-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]pyridine-2-carboxamide
4-[2-(2-aminopyrimidin-5-yl)-7,8-dimethylquinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
4-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,2,5-oxadiazole-3-carboxamide
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]propanamide
2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyridine-4-carboxylic acid
6-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]pyridine-2-carboxylic acid
2-(2-chlorophenyl)-3-methyl-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(furan-3-ylmethyl)-4-hydroxy-N-methyl-2-phenylpyrimidine-5-carboxamide
1-(3,5-dimethylbenzoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylic acid
4-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(1-{imidazo[1,2-a]pyridine-6-carbonyl}azetidin-3-yl)pyridine
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-9H-purin-6-amine
1-(4-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
3-(cyclohex-1-en-1-yl)-5-[(oxolan-2-ylmethyl)sulfamoyl]benzoic acid
1-{[1-(2,3-dihydro-1H-inden-4-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]piperidine-1-carbonyl}pyridine
(3S,4S)-4-[(adamantan-1-ylmethyl)(methyl)amino]-1-(benzenesulfonyl)pyrrolidin-3-ol
3-hydroxy-3-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-{[2-(benzyloxy)phenyl]methyl}-1,1-dioxo-1λ6-thiolane-3-carboxamide
3-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-N-(1,3,4-thiadiazol-2-yl)benzamide
N-cycloheptyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
methyl 3-{[(1-phenylcyclohexyl)formamido]methyl}-5-(pyrazine-2-amido)benzoate
8-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-4-amino-1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
4-{3-[(3S)-3-(dimethylamino)azepane-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
1-(methoxymethyl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-(4-fluorophenyl)-3-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
5-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]pentanoic acid
2-[4-({cyclopropyl[(2-ethoxyphenyl)methyl]carbamoyl}amino)phenyl]-N-methylacetamide
3-chloro-N-[4-(4-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
5-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(3-methoxyphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(1,3-dihydro-2-benzofuran-5-yl)urea
4-{[3-(2-aminoethyl)phenyl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
2-{4-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]phenoxymethyl}pyridine
N,N,6,8-tetramethyl-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
8-(quinolin-2-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
3-hydroxy-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol