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2-ethyl-9-(2-methyl-1H-pyrrole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
(4aR,7aS)-1-butyl-4-(2-chloro-5-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(furan-3-yl)-1-(4-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-methoxypyridine
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(benzyloxy)-3-chlorophenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-hydroxy-5-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}benzoic acid
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-2-(methylsulfanyl)ethan-1-one
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(1H-pyrazol-1-yl)butan-1-one
2-[2-(4-methoxybenzoyl)-1H-imidazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
7-(cyclopropylmethyl)-2-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-(pyridine-3-carbonyl)piperidin-4-amine
3-cyclohexyl-N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
9-[2-(3-hydroxypiperidin-1-yl)acetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[(diethylamino)methyl]-N-[4-(propan-2-yl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-methyl-N-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]propanamide
N-(2-hydroxyethyl)-3-methyl-N-(thiophen-2-ylmethyl)furan-2-carboxamide
N-benzyl-2-(pyrrolidin-3-yl)-N-(2,2,2-trifluoroethyl)acetamide
1-[(6-methylquinolin-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(3,5-difluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(quinolin-2-ylmethyl)-1,4-diazepan-5-one
2-[(4-cyanopiperidin-1-yl)methyl]-3,5-dimethoxybenzoic acid
3-({2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1λ6-thiane-1,1-dione
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
11-(4-ethylpiperazin-1-yl)-4-(3-methylbutyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2S,4R)-4-amino-1-(2,8-dimethylquinoline-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrazine
4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-phenylpiperazin-2-one
3-(4-methyl-1,3-thiazol-5-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
[(3R,4R)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
(3S)-3-{[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}azepan-2-one
benzyl(butyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
(2S,4S)-N-ethyl-4-[2-(thiophen-2-yl)acetamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
2-(5-fluoro-2-methylphenyl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
N-[4-(furan-2-ylmethoxy)phenyl]-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][(2-phenyl-1,3-oxazol-4-yl)methyl]amine
{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N,N-diethyl-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]benzamide
3-(thiomorpholine-4-carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
5-(2-ethoxyphenyl)-1H-indazole
2-(3-methoxyphenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N'-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N'-(oxolan-2-ylmethyl)ethanediamide
3-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carbonitrile
6-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-2-methyl-2,3-dihydropyridazin-3-one
8-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(2R,6R)-4-[2-(cycloheptylcarbamoyl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
6-ethyl-1,5-dimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide