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3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-{[1-(cyclopropylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperidin-4-yl)acetamide
1-[5-cyclopentyl-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
2-(3-methoxypropyl)-1-(naphthalene-1-carbonyl)piperidine
(4aS,8aR)-6-(3-chloropyridin-2-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
1-ethyl-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[4-(2-methoxyethoxy)phenyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetic acid
5-[4-(trifluoromethyl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinoline
3-[(methylsulfanyl)methyl]-5-[1-(2-phenylethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
3-[N-benzyl-2-(2,3-dihydro-1H-inden-1-yl)acetamido]propanamide
1-(2-methyl-1-benzofuran-5-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
2-(3-fluorophenyl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]ethan-1-one
1-ethyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methyl-1H-pyrazole-3-carboxamide
5-(1H-indol-1-ylmethyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
2-(3-hydroxyphenyl)-2-[4-(4-methoxybenzoyl)piperazin-1-yl]acetic acid
(1R,3S)-3-ethoxy-7-(2-propyl-1,3-thiazole-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(2S)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(2S)-2-{[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]amino}-3-(1H-indol-3-yl)propan-1-ol
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
3-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]benzamide
3-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-[(4-chlorophenyl)methyl]-8-(6-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine-1-sulfonamide
1-{2-hydroxy-3-[3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
3-hydroxy-1-(2-phenylethyl)-3-({[2-(1H-pyrrol-1-yl)ethyl]amino}methyl)piperidin-2-one
1'-(1-methyl-1H-imidazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-ethyl-8-methyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-2-(morpholin-4-yl)-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,3-benzodiazole
(3S,4R)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoacetamide
(1S,5R)-6-[(1-ethyl-1H-indol-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4-methoxyphenyl)methyl]-4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
5-cyclopropyl-N-[2-(pyridin-3-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-cyclohexyl-N3-[2-(3-methoxyphenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-methyl-1,3-thiazol-4-yl)-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-(2-methylpropyl)-2-(morpholin-4-yl)-N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)acetamide
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-{[4-(methylsulfanyl)phenyl]methyl}cyclopropanamine
5-fluoro-N-methyl-2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-1-phenylmethanesulfonamide
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-4-yl)propan-1-one
5-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methoxyethan-1-one
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide