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1'-(2,3-dihydro-1-benzothiophene-2-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-methyl-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
(4aS,7aR)-1-(2-hydroxyacetyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-ethyl-4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[5-(4,5-dimethylthiophen-2-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
4-methyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]-1,3-oxazole-5-carboxamide
(1R,3S,5S)-3-({1-[1-(4-methylpyridin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methoxy)-8-azabicyclo[3.2.1]octane
4-(2,6-dimethoxypyrimidin-4-yl)benzoic acid
3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}azetidin-3-yl)pyridine
1-[(5-methylfuran-2-yl)methyl]-N3-[(2-methylphenyl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine
dimethyl(3-{2-[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
6-{[2-(1,3-thiazol-4-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
(1R,3S)-7-(2,6-dimethylpyrimidine-4-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N5-cyclooctyl-N3-(furan-2-ylmethyl)-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[1-(cyclohex-1-en-1-yl)ethyl]acetamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(1R,3S)-3-amino-N-[(5-fluoro-2-methylphenyl)methyl]cyclohexane-1-carboxamide
2-{[6-(2-chloro-4-fluorophenyl)pyridazin-3-yl]amino}ethan-1-ol
2-ethyl-9-[2-(morpholin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
2-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2-oxazinane
N3-cyclooctyl-N5-(furan-2-ylmethyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]acetic acid
N-methyl-N-(oxan-2-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
1-[(3,4-dimethylphenyl)methyl]-4-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperazin-2-one
N,7-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-cyclopropyl-1-[1-(2-fluorobenzoyl)piperidin-4-yl]piperidine-3-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclopent-1-ene-1-carboxamide
1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
4-(3-fluorophenoxy)-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxylic acid
(3R,4S)-3,4-dimethyl-1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperidin-4-ol
1-({3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
1-(propan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
5-(9H-purin-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}-5-methoxy-1,4-dihydropyridin-4-one
5-(methoxymethyl)-3-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,2,4-oxadiazole
5-ethyl-N4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrimidine-2,4-diamine
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(morpholin-4-yl)ethyl]propanamide
4-({4-methyl-5-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
9-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
[1-(benzenesulfonyl)-3-propylpiperidin-3-yl]methanol