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2-[(3-fluorophenyl)methyl]-6-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(3R,4S)-4-(4-methoxyphenyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-amine
6-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-9H-purin-2-amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-[1-hydroxy-3-(methylsulfanyl)propyl]-1H-1,2,4-triazol-3-yl]acetamide
1-[1-(8-methoxyquinolin-2-yl)piperidin-4-yl]piperidin-4-ol
8-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
1-[2-(4-chloro-3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-3-ol
1-{2-[1-(1,3-benzothiazole-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
1-({4-methyl-5-[1-(pyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
7-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylate
1-methyl-2-oxo-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(1-methyl-1H-pyrazol-5-yl)propanamide
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-2,7,8-trimethylquinoline-4-carboxamide
4-hydroxy-2-methyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
methyl[2-methyl-2-(piperidin-1-yl)propyl][1-(pyrazin-2-yl)propan-2-yl]amine
N-cyclopropyl-1-{1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-4-yl}piperidine-3-carboxamide
1-(2,5-difluorophenyl)-3-[2-(propan-2-ylsulfanyl)ethyl]urea
4-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperazine-1-carboxamide
N1,N1-dimethyl-N4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine-1,4-dicarboxamide
6-propyl-2-(2-{[2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]-N-methylbutanamide
2-(9H-carbazol-3-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
N'-cyclopentyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)butanediamide
2-(2-chlorophenyl)-N-(2-methoxy-2-methylpropyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-cyclopentyl-3-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]propanamide
1-ethyl-3-[2-(2-fluorophenoxy)pyridin-3-yl]-1-(oxan-2-ylmethyl)urea
6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]hexan-1-ol
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
2,5,6-trimethyl-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]pyrimidin-4-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6-methylquinolin-3-yl]methyl}cyclohexanecarboxamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
4-ethyl-1-methyl-3-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-(4-chlorophenyl)-4-(4-methyl-1H-imidazole-5-carbonyl)morpholine
7-methyl-2-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[2-(4-phenylpyrimidin-2-yl)ethyl]amine
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]propanamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-amino-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-phenylpyrimidine-5-carboxamide
2-hydroxy-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(3aS,6aS)-2-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
dimethyl({2-[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-(3-methylthiophen-2-yl)ethyl})amine
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperidine
1-{3-[4-({[(2-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
6-{[(1S,2S)-2-hydroxycyclohexyl]amino}-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide