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N-[2-(4-chlorophenyl)-2-(piperidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
1-[2-({7-methanesulfonyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]imidazolidin-2-one
3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]-1-(thiophen-2-ylmethyl)piperidine
3-methyl-7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-cyclopropyl-6-(1H-indol-4-yl)pyridazin-3-amine
5-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(5-methylthiophen-2-yl)-4-(piperidin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(5-chlorothiophene-2-carbonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
1-ethyl-8-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(oxan-2-yl)ethyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-[1-benzyl-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
4-methyl-2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]quinazoline
N-(2,2-dimethylpropyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[3-(3-methoxyphenyl)phenyl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidine-2-carboxamide
2-[3-(1,3-dimethyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2-fluoro-6-methoxybenzoyl)piperidine
N-methyl-4-[4-(piperidin-1-ylmethyl)phenyl]benzene-1-sulfonamide
N-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)acetamide
5-butyl-4-methyl-6-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]pyrimidin-2-amine
ethyl 2-(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
N-ethyl-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-ethyl-3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}propanamide
2-{[3-(2-carbamoylethyl)piperidin-1-yl]methyl}benzoic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
1-[4-(pyridin-4-yl)piperidin-1-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-3-methoxypyrazine
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-cyclopentanecarbonyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]piperidine-4-carboxamide
N-[3-(4-ethoxyphenyl)propyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethyl-8-(4-hydroxy-3-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(2,3-dihydro-1H-inden-2-yl)azetidin-3-yl]-2-methylpiperidine
3-methoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazin-2-amine
3-[3-cyclopropyl-5-(7-fluoro-3-methyl-1H-indol-2-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dimethylquinoxaline-6-carboxamide
6-(methoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidin-4-amine
2-cyclopropyl-5-[2-(4-methylpentyl)morpholine-4-carbonyl]-3,4-dihydropyrimidin-4-one
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
2-{1-ethyl-5-[5-(ethylsulfanyl)thiophen-2-yl]-1H-1,2,4-triazol-3-yl}acetamide
N-[(3R,4S)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
2-[4-(2-methanesulfonylethyl)piperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
(3aS,6aR)-5-(1-ethylpiperidin-4-yl)-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methyl-6-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]pyrimidin-4-ol
N-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)pyridin-3-amine
3-methyl-5-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-[(2-methylpyrrolidin-1-yl)methyl]-1,3-oxazole
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide