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1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(2-methyl-1-benzofuran-5-yl)urea
(3-{[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
ethyl 1-(1H-imidazol-2-ylmethyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}thian-4-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
{4-[6-(propan-2-yl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
4-(1,6-naphthyridin-5-yl)phenol
ethyl 3-[(3-chlorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylate
3-(methylsulfanyl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(azepan-1-yl)-3-[3-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1-(propan-2-yl)-1H-pyrrole-2-carboxamide
1-(3-ethylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
(2H-1,3-benzodioxol-5-ylmethyl)(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
8-(2,3-dihydro-1H-inden-2-yl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[3-methyl-7-(thiophene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenoxypropanamide
N-[4-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)phenyl]acetamide
6-ethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
9-(pyrimidin-5-ylmethyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-(dimethylamino)-1-(4-phenoxybenzoyl)pyrrolidine-2-carboxylic acid
(5-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
3-chloro-4-({1-[(3-chlorophenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-[(2-hydroxyethyl)({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
4-[2-(4-chlorophenyl)-2-hydroxyacetyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
[(5-ethylfuran-2-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
3-[3-(aminomethyl)phenyl]-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
ethyl 4-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]piperidine-1-carboxylate
4-amino-2-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]pyrimidine-5-carbonitrile
2-[1'-(1-ethyl-1H-pyrazole-4-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
7-(cyclohexylmethyl)-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
3-(2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-3-phenylprop-2-yn-1-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
8-methoxy-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}pyridin-3-ol
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
(3R,5S)-5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-3-ol
1-tert-butyl-5-oxo-N-[2-(1,3-thiazol-4-yl)ethyl]pyrrolidine-3-carboxamide
6-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrimidine-2,4-diamine
2-(propan-2-yl)-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-tert-butyl-4-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidin-2-one
1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]thiophene-2-carboxamide