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6-[1-(1-cyclohexylpiperidine-4-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-ethyl-N-methyl-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-sulfonamide
4-[(2-ethoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
5-chloro-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-(trifluoromethyl)pyridin-2-amine
N-methyl-N-(propan-2-yl)-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
1-[6-hydroxy-4-(oxan-4-yl)-1,4-diazepan-1-yl]-2-(4H-1,2,4-triazol-4-yl)ethan-1-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(2H-1,3-benzodioxol-5-yl)-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-ethyl-2-{[2-(pyridin-3-yl)quinolin-4-yl]formamido}propanamide
1-(4-{[4-({4-[methyl(phenyl)amino]phenyl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
2-(2-chloro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenoxy)propanoic acid
[(8-methoxyquinolin-2-yl)methyl](methyl)(oxan-2-ylmethyl)amine
2-methylpropyl (2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(1R,5S,6R,7S)-6-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}-3-(propan-2-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]benzamide
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(1S,5R)-3-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
2-(methylsulfanyl)-5-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidine
4-{[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-N,N,1-trimethylpiperidin-4-amine
6-{1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]piperidin-3-yl}-2-methylpyrimidin-4-ol
3-({1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
3-chloro-5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(azocan-1-yl)-3-{2-methoxy-4-[(methylamino)methyl]phenoxy}propan-2-ol
4-[2-(4-fluorophenoxy)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-ethyl-4-phenyl-9-(1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecane
1-[cyclohexyl(methyl)amino]-3-(2-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
4-{1-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-2-methyl-3-oxo-4-phenylpiperazine-1-carboxamide
1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-(1H-pyrazol-4-yl)butanamide
4-ethyl-3-{[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(piperazin-1-yl)ethyl]-N-[2-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-(1-benzofuran-2-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-(furan-3-ylmethyl)-N,2-dimethylthieno[2,3-d]pyrimidin-4-amine
2-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4H-chromen-4-one
2-(ethylamino)-N-(thiolan-3-yl)pyrimidine-5-carboxamide
3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-1H-indazole
2-(dimethylamino)-2-(3-methylphenyl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)acetamide
2-(3,5-dimethoxyphenyl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
N-cyclopropyl-5-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-{1-[(5-chlorofuran-2-yl)methyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
N-[2-(1H-indol-3-yl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
1-(4-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one