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{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(thiophen-3-ylmethyl)amine
4'-[2-(2-methoxyphenoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1S,5R)-3-(1-ethyl-1H-pyrazole-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(cyclohex-1-en-1-yl)ethan-1-one
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(9H-purin-6-yl)piperidin-4-amine
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}naphthalen-1-ol
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
{[(3R,4S)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}(ethyl)methylamine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)acetamide
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(pyrimidin-2-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
8-(1-methanesulfonylpropan-2-yl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)-N-[1-(pyridin-2-yl)propyl]acetamide
{1-[2-(1H-pyrazol-1-yl)ethyl]piperidin-4-yl}(thiophen-2-yl)methanol
5-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-phenyl-1,2-oxazole
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-1-methyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-2-ynamide
5-methoxy-1-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-indole-2-carboxamide
3-(2-methoxyethyl)-6-methyl-3,4-dihydroquinazolin-4-one
(4aS,8aR)-1-(2-methylpropyl)-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methylacetamide
4-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
(4aS,8aR)-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{4-[2-(3-ethoxy-4-hydroxyphenyl)-1H-imidazol-1-yl]phenyl}acetamide
{3-[(8-methylquinolin-5-yl)methyl]-9-(propan-2-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
5-cyclopropyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1,3,4-oxadiazol-2-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}benzamide
(1R,6S)-9-methyl-3-[2-(1H-pyrazol-1-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[(2-methylphenyl)(phenyl)methyl]-2-(pyridin-4-yl)acetamide
7-[(4-fluorophenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-cyclopropanecarbonyl-1'-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-5,6-dimethylpyridine-3-carbonitrile
6-chloro-N,N-dimethyl-3-(morpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
(3aR,6aS)-5-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-phenyl-5-[(3,4,5-trifluorophenyl)methyl]-1H-1,2,4-triazole
3-(1-cyclopropanecarbonylpiperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-{4-[4-(pyridin-4-yl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-2-(6-methoxypyridin-3-yl)acetic acid
3-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1-(2-methylphenyl)urea
(3S,5R)-N3-(2-acetamidoethyl)-N5-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(pyrrolidin-1-yl)acetamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-(furan-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-(2-hydroxyethyl)-9-[(3,4,5-trifluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one