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(3R,5S)-N-butyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(6-methoxypyridin-3-yl)methyl]methylamine
methyl 4-{[9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
N-{1-[3-(2-chlorophenoxy)azetidin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
(4aS,8aS)-2-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-decahydroisoquinolin-4a-ol
N-(1-benzylpyrrolidin-3-yl)-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
(1S,5R)-6-[(2-fluoro-5-methylphenyl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(3-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-(3-fluorophenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-{2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-(butan-2-yl)-2-(ethylamino)-4-methyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-5-carboxamide
ethyl 1-[(2,4-dimethylphenyl)carbamoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-{4-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(4-methyl-1,4-diazepan-1-yl)butan-1-one
2-amino-6-(4-hydroxy-3-methoxyphenyl)-4-(quinolin-5-yl)pyridine-3-carbonitrile
4-(4-methylphenoxy)-1-(oxane-2-carbonyl)piperidine-4-carboxylic acid
1-(azepan-1-yl)-3-[3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(4-methoxy-2-methylphenyl)-3-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]propanamide
2-[(3,5-dimethoxyphenyl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-ethoxy-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(prop-2-en-1-yloxy)-N-(propan-2-yl)benzamide
3-methyl-4-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-3,4-dihydroquinazoline-7-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-{3-phenyl-3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(2-hydroxyethyl)piperidine-4-carboxamide
(8R,9aS)-2-{[1-(ethoxymethyl)cyclobutyl]methyl}-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
3-(carbamoylamino)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]propanamide
5-acetyl-N-[2-(3-chlorophenyl)ethyl]thiophene-3-carboxamide
(4aR,7aS)-6,6-dioxo-N-(4-oxo-4H-chromen-6-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(4-methoxyphenyl)methyl]-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
2-{4-[1-(dimethylamino)ethyl]phenyl}-N-ethylpyrimidin-4-amine
1-benzyl-4-(1H-indazole-3-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
13-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-4-methyl-2-phenyl-1,3-thiazole
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N,N,7,8-tetramethylquinoline-4-carboxamide
8-[(6-chloropyridin-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]acetamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)[(5-ethylpyridin-2-yl)methyl]methylamine
(4aS,7aR)-1-(3-methoxy-4-methylbenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-acetyl-N-[2-(1H-imidazol-4-yl)ethyl]thiophene-3-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-{[1-(pyridin-2-yl)propyl]amino}pyridine-3-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxane-4-carbonyl)piperidine