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2-[5-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyridine
11-{[(2,6-difluoro-3-methylphenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(4-ethylpiperazin-1-yl)-N-(2-phenylethyl)-2,3-dihydro-1H-indene-2-carboxamide
methyl 2-{[6-amino-2-(diethylamino)pyrimidin-4-yl](methyl)amino}acetate
1-{[4-(2-fluorophenyl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
5-(2-fluorophenoxymethyl)-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
2-[4-(isoquinolin-5-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
2-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxy-4H-pyran-4-one
(1R,3S)-3-(2-aminoethoxy)-7-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-7-azaspiro[3.5]nonan-1-ol
(4aR,8aS)-6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-(4-fluorophenyl)-4-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
1-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
3-(2-fluorophenyl)-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)propanamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]propanamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[2-(pyrrolidin-1-yl)phenyl]propanamide
5-{3-[4-(4-fluorophenoxy)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
1-[(3,4-difluorophenyl)methyl]-3-(2,4-dimethoxybenzoyl)piperidine
N-(2,1,3-benzothiadiazol-4-yl)-4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carboxamide
(2S)-1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-N-ethylpyrrolidine-2-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}benzamide
1-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)azepan-2-one
5-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(3-methylphenyl)pyrimidine
N-(3-fluoro-2-methylphenyl)-3-propylmorpholine-4-carboxamide
methyl({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
5-{2-[1-benzyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethylpyrimidin-2-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[1-(1H-imidazol-2-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
N-cyclopropyl-1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
2-chloro-5-{[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}pyridine
1-[(4-fluorophenyl)methyl]-5-(2-methoxybutanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-ethylpiperidin-4-yl)piperidine
1-(4,6-dimethylpyrimidin-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
3-[(4-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}piperidin-1-yl)methyl]pyridine
3-ethyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-[4-(1H-pyrazol-5-yl)phenyl]urea
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
4-hydroxy-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
3-methyl-4-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-(2-methylpropyl)piperazin-2-one
N,N-dimethyl-6-{3-oxa-9-azaspiro[5.5]undecan-9-yl}pyrazine-2-carboxamide
1-(2-chlorophenyl)-4-(2-hydroxy-4-methylbenzoyl)piperazin-2-one
8-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
2-ethoxy-5-{2-[(1-methylpiperidin-4-yl)amino]pyrimidin-4-yl}benzoic acid
1-(cyclohexylmethyl)-5-(ethylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})(quinolin-4-ylmethyl)amine