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1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-methoxyphenyl)ethan-1-one
6-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2,3-dihydropyridazin-3-one
N-(3,4-dimethoxyphenyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-amine
3-methyl-8-[2-(1H-pyrazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(S)-(2-chlorophenyl)[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methanamine
3-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
(2S,4S)-N-methyl-4-[4-(4-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
4-ethyl-1-methyl-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
3-{4-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]piperazin-1-yl}benzoic acid
4-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(3-methyloxetan-3-yl)methyl]acetamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(2-methylfuran-3-carbonyl)piperidin-3-amine
4-(hydroxymethyl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)azepan-4-ol
3-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
3-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-(2,6-dichloropyridin-4-yl)-8-methyl-2,8-diazaspiro[4.5]decane-2-carboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(1-benzofuran-2-yl)-4-(5-methyl-1H-imidazol-2-yl)-1H-pyrazole
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]-N-(propan-2-yl)quinoline-4-carboxamide
3-[2-(adamantan-1-yl)acetamido]-4,4,4-trifluorobutanoic acid
methyl 3-(4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3-dihydropyridazin-3-one
N-{4-methyl-2-[3-(pyridin-3-yl)propanamido]phenyl}benzamide
5-methyl-3-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-ethylpyrimidine-5-carboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-{4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}-1-ethylpyrrolidin-2-one
4-[(4-{2-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-4-methylphenoxy}piperidin-1-yl)methyl]pyridine
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
3-{2-oxo-2-[3-(4-phenylbenzoyl)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
2-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-ethyl-1-[4-(propylsulfamoyl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
({4-[(3,5-dichloro-2-methoxyphenyl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
2-chloro-4-({[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-6-methoxyphenol
2-chloro-N-({1-[(3S,5S)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)pyridine-4-carboxamide
6-methoxy-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrimidin-4-amine
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3,3-diphenylpiperidine
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(2-aminoethyl)-N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-[2-(1-ethylpiperidin-4-yl)acetyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
7-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
3-cyclopropyl-1-{4-[5-(morpholine-4-carbonyl)furan-2-yl]phenyl}urea
4-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid