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9-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[3-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}methoxy)phenyl]propanamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2-phenyl-1H-imidazol-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
2-methyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-6-(piperidin-4-yl)pyrimidin-4-amine
2-benzyl-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-(4-{1-[(tert-butylcarbamoyl)amino]cyclohexyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-(furan-2-yl)-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]azepane
2-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]thiophene-3-sulfonamide
N-[2-(2-fluorophenyl)ethyl]-5-{4-hydroxy-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
5-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-yl)-2-phenyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-{4-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]thiophen-2-yl}ethan-1-one
N-(2-oxoazepan-3-yl)-2-propyl-1,3-thiazole-4-carboxamide
8-(4-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)quinoline
2-{5-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
3-(difluoromethoxy)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
2,5-dioxo-6-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[(pyridin-3-ylmethyl)sulfamoyl]-N-(pyrimidin-4-ylmethyl)benzamide
5-propyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-3-carboxamide
3-{4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
(3S,4R)-1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
4-(4-methyl-1H-pyrazol-1-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine-4-carboxylic acid
1-[(4-fluoro-3-methoxyphenyl)methyl]-N-(4-fluorophenyl)piperidin-3-amine
2-[2-(azepan-1-yl)ethyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
4-({4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)piperidine
2-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,4-dihydroquinolin-4-one
3-(3,5-dimethylphenyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}propanamide
3-(3-fluorophenyl)-1-[4-(pyridin-3-yl)piperazin-1-yl]propan-1-one
5-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridine-2-carbonitrile
5-(2-fluorophenyl)-N-(2-methoxybutyl)pyrazolo[1,5-a]pyrimidin-7-amine
(1R,5R)-3-{pyrazolo[1,5-a]pyridine-3-carbonyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-benzothiophen-2-ylmethyl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N'-(2,3-dimethylphenyl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}propanediamide
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)azepane
3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3,9-diazaspiro[5.6]dodecan-10-one
3-{2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
5-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}amino)acetate
1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-5-(5-cyclopropyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole
4-[(dimethyl-1,3-thiazol-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-benzyl-5-{[propyl(pyridin-3-ylmethyl)amino]methyl}pyrimidin-2-amine
1-{1-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]piperidin-3-yl}pyrrolidin-2-one
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
5-methyl-1-[4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole