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N-(2-hydroxy-1-phenylethyl)-4-(4-methylphenoxy)piperidine-4-carboxamide
3-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)carbamoyl]amino}phenyl)-N,N-dimethylpropanamide
2-(1-ethylpiperidin-4-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)acetamide
N-(4-{2-[methyl(pyridin-2-ylmethyl)amino]acetamido}phenyl)pentanamide
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
1-(furan-2-ylmethyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(dimethyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
3-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-pyrazole
2-(5-{1-[2-(pyrimidin-2-yl)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
3-hydroxy-2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-(pyridin-2-ylmethyl)piperazine
9-(2-ethoxypropanoyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-{3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxybenzoyl}piperidin-3-yl)propan-1-one
1-(3-methylpyridin-4-yl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
2-ethyl-N-(2-phenylethyl)-2H-1,2,3,4-tetrazol-5-amine
methyl 2-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}-1,3-oxazole-4-carboxylate
3-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-(2-methoxy-5-{[methyl(thian-4-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
(3R,4R)-1-(3-cyclopentylpropyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-({5-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
(3R,4S)-4-cyclopropyl-1-(7-fluoro-4-methylquinolin-2-yl)pyrrolidin-3-amine
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[3-(pyrrolidin-1-yl)propyl]-1H-imidazole
5-[(R)-methoxy(phenyl)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
2-(1H-1,3-benzodiazol-1-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[(2-benzylmorpholin-4-yl)methyl]-2-methoxy-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-methyl-1-{3-[4-(3-methylphenyl)piperazin-1-yl]propanoyl}-1,4-diazepan-5-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-chloro-N-{1-[1-(3-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-(2,6-dimethylpyridin-3-yl)-1-[(2-methylphenyl)methyl]-1-(oxolan-2-ylmethyl)urea
1-benzyl-4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-5-methyl-1H-1,2,3-triazole
1-methyl-N-[(3-methylpyridin-2-yl)methyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(3-cyano-4-methoxyphenyl)-4-(thian-4-yl)piperazine-1-carboxamide
3-(morpholine-4-sulfonyl)-5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]benzoic acid
2-{[5-(furan-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-{[(1-ethylpiperidin-4-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
methyl 6-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}pyridine-2-carboxylate
2-amino-N-[(2-chlorophenyl)methyl]-N-cyclopropyl-4-phenylpyrimidine-5-carboxamide
N'1-[(3R,4S)-1-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
methyl (2S,4R)-1-methyl-4-[1-(3-methylbutanoyl)piperidine-4-amido]pyrrolidine-2-carboxylate
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-(quinolin-8-yl)piperidine-1-carboxamide
N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methoxypyridin-3-yl)urea
(1R,7S)-3-(2-ethylbutyl)-6-[3-(morpholin-4-yl)azetidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(dimethylamino)-2-(2-methylphenyl)-N-(1-propylcyclopropyl)acetamide
N-[(3,4-difluorophenyl)methyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide