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4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
6-(aminomethyl)-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
1-{2-[4-(cyclohex-3-en-1-ylmethyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-[(3-methoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]morpholine
1-{3-oxo-3-[3-(pyridin-2-yl)azetidin-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(1-benzyl-4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}piperazin-2-yl)ethan-1-ol
{1-[3-(trifluoromethyl)benzenesulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]quinoline-8-sulfonamide
1-(4-amino-5-cyanopyrimidin-2-yl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-(3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
[(1R,3S,3aS,6aR)-5-methyl-1-(2-methylpropyl)-3-(5-methylthiophen-2-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-(2,2-diphenylethyl)-N-methylpiperidine-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
[(3S,5R)-1-(3,5-difluoro-4-methoxybenzoyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[3-(2-methylphenyl)phenyl]methyl}amine
N,N-dimethyl-2-[2-(4-methylpiperazin-1-yl)pyrimidin-5-yl]quinoline-4-carboxamide
5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(2-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
1-{1-[1-(thiolan-3-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}cyclopentan-1-ol
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4R)-1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4-phenylpyrrolidine-3-carboxylic acid
1-[5-(dimethylcarbamoyl)pyridin-2-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
methyl (2S)-3-methyl-2-[(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazol-3-yl)formamido]butanoate
3-cyclohexyl-N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-1H-pyrazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxy-4-methylbenzamide
4-(benzyloxy)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
2-(adamantan-1-yl)-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)acetamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]acetamide
1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}azepane
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,5-dimethyl-1H-indole-2-carboxamide
1-(4-{[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(2R)-2-{[4-(4-methoxyphenoxy)phenyl]formamido}-3-methylbutanamide
1-(4-{2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-methylpropan-1-one
N-(2-hydroxyethyl)-1-(oxan-4-yl)-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-(furan-3-ylmethyl)-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
1-(furan-3-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
6-(2-methoxyphenyl)-N-[(2-methylphenyl)methyl]pyridazin-3-amine
1-[3-methoxy-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole
1-{2-[methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})amino]ethyl}piperidin-2-one
N-(2-hydroxyethyl)-2-(phenylamino)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}piperidin-3-ol
2-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-ethoxyphenol
dimethyl[(4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-thiazol-2-yl)methyl]amine
methyl 4-{[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]carbamoyl}piperazine-1-carboxylate
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
1-(3-cyclopentylpropanoyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-(4-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one