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5-(methoxymethyl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
7-(1H-indol-2-ylmethyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-benzyl-4-[5-(methoxymethyl)thiophene-2-carbonyl]piperazin-2-one
4-[(4-hydroxyphenyl)methyl]-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
8-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
5-(4-fluorophenyl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-methyl-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
{[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}urea
(1s,4s)-4-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)cyclohexan-1-amine
1-[(4-methoxyphenyl)methyl]-4-(3-methoxypropanoyl)piperazin-2-one
2-[(1R,3S,3aS,6aR)-1-(hydroxymethyl)-5-methyl-3-[5-(4-methylphenyl)furan-2-yl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
1-{[4-methyl-5-(1-pentylpiperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
4-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-1-(4-methoxyphenyl)piperazin-2-one
2-(2-methoxyethyl)-9-[2-(3-methoxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-[5-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-[(3R,4S)-4-cyclopropyl-1-(2-methylpyridin-4-yl)pyrrolidin-3-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1-(3,5-dimethylphenyl)piperazin-2-one
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-{[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
(3S,4R)-1-[3-(difluoromethoxy)benzoyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
5-[4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2,5-dimethylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-(4-fluoro-2-methoxyphenyl)-3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
(2S)-1-[3-(azocan-1-yl)propanoyl]-N,N-dimethylpyrrolidine-2-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})(oxolan-2-ylmethyl)amine
1-[(3-methoxyphenyl)methyl]-4-(5-methylthiophene-3-carbonyl)piperazin-2-one
3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}oxolane-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]pyrimidin-2-amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-{[1-(9H-purin-6-yl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
1-{1-[(4,5-dimethylfuran-2-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
3-[(3R,4S)-1-(1-benzofuran-5-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[(1-{1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
3-({4-[2-(1H-imidazol-1-yl)ethyl]piperazin-1-yl}methyl)-8-methyl-1,2-dihydroquinolin-2-one
methyl 8-[(2E)-2-methylbut-2-en-1-yl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-cyclopropyl-2-[4-({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidin-1-yl]acetamide
1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
(3S,4R)-1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-[(5-chloro-2,4-dimethoxyphenyl)methyl]-1-methylpiperazine-2-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2,5-dimethoxyphenyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}acetamide
N-methyl-5-(phenoxymethyl)-N-(quinolin-3-ylmethyl)-1H-pyrazole-3-carboxamide
3-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
methyl({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})(quinoxalin-6-ylmethyl)amine
methyl (2S)-2-{[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]amino}-3-phenylpropanoate
9-[(3-methyl-1-benzofuran-2-yl)methyl]-3-oxa-9-azaspiro[5.5]undecane