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(1R,3S)-N-(2H-1,3-benzodioxol-5-yl)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-[2-(pyrazin-2-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
8-[(2E)-but-2-en-1-yl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(1-acetylpiperidine-3-carbonyl)piperazin-1-yl]-N-(pyridin-3-yl)acetamide
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-{4-[3-(2-aminoethyl)phenyl]phenyl}methanesulfonamide
1-[2-fluoro-6-(trifluoromethyl)phenyl]-3-(5-hydroxypentyl)urea
1-{1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carbonyl}-1,4-diazepane-6-carboxylic acid
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-5-(cyclobutylmethoxy)benzoic acid
(1R,9aR)-1-({[(2,4-dimethoxyphenyl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-2-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N3-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
5-acetyl-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]thiophene-2-carboxamide
3-cyclopropyl-5-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)-1H-1,2,4-triazole
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
N-(1-methyl-1H-pyrazol-3-yl)-2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]acetamide
2-(3-hydroxypropyl)-9-[2-(methylsulfanyl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4H-thieno[3,2-b]pyrrole-5-carboxamide
7-(1,2,3,6-tetrahydropyridin-1-ylmethyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(oxan-4-yl)piperazine
8-(5-chloro-2-methoxybenzenesulfonyl)-2,8-diazaspiro[4.5]decan-3-one
1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
5-chloro-4,6-dimethyl-3-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-methyl-N-(2-methylpropyl)-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
2-[(4,6-dimethylpyrimidin-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(2E)-N-{[7-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
(3S,4S)-1-[1-(4-methoxyphenyl)piperidin-4-yl]-4-methylpiperidine-3,4-diol
1-(2,6-difluorobenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-[(dimethyl-1,2-oxazol-4-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methoxybenzoyl)piperazine
1-[2-({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,2-dione
1'-[(5-methylthiophen-2-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(quinoxalin-5-ylmethyl)piperidin-3-yl]propanamide
6-methyl-2-(3-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-(1,3-benzothiazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)azepan-2-one
1-benzoyl-4-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperazine
6-ethoxy-3-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]pyrrolidine-2-carboxylic acid
3-cyclopropyl-1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperazine
1-ethyl-N-(3-phenylpropyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(diethylamino)ethyl]-1H-pyrazole-4-carboxamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-oxo-1,6-dihydropyridazine-3-carboxamide