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1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-tert-butyl-3-[(3,4-dimethoxyphenyl)methyl]-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-({[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]amino}methyl)-N-methylfuran-2-carboxamide
6-[(diethylamino)methyl]-N-(1-hydroxypropan-2-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(1H-pyrazol-1-yl)-1-(thiophen-3-ylmethyl)piperidine-4-carboxylic acid
2-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
2-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]pyridin-3-ol
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-2-(4-phenylphenyl)acetamide
3-(4-fluorophenyl)-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
5-[2,6-dimethyl-4-(pyrrolidin-1-ylmethyl)phenoxy]-1-azabicyclo[3.2.1]octane
4-benzyl-1-(thiolan-3-yl)piperidine
6-methyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
1,3-dimethyl-4-[(1-{[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
2-(2-chloro-5-methylphenyl)-2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]acetic acid
1-methyl-4-[2-(3-methyl-4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)ethyl]piperazine
1-{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
3-[(2-fluorophenyl)methyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
8-(2-ethoxyethyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1s,4s)-4-(4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)cyclohexan-1-amine
methyl[1-(pyridin-3-yl)ethyl]{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
3-[(3R,4S)-1-[2-(dimethylamino)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
5-(azocane-1-carbonyl)-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-(1-{[1-(thiolan-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)cyclopentan-1-ol
2-(2-{2-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)pyrazine
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
1-({3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}methyl)-4-(pyridin-2-yl)piperidin-4-ol
(1S,9R)-11-[3-(1,2-oxazinan-2-yl)propanoyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-amino-8-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
(3R,5S)-5-(pyrrolidine-1-carbonyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
(2S)-2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-phenylpropan-1-ol
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-(3,5-dimethyl-1-{[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazol-4-yl)ethan-1-one
N-(2-methanesulfonylethyl)-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-N-(propan-2-yl)pyrimidin-4-amine
N-(2,4-dimethoxyphenyl)-3-[1-(oxan-4-yl)piperidin-4-yl]propanamide
(cyclohex-3-en-1-ylmethyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylpyridine-3-carboxamide
2-{3-oxo-9-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-methoxy-1-{4-[4-(thiomorpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
7-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)-4-methyl-2H-chromen-2-one
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-methyl-N-(propan-2-yl)acetamide
3-[2-fluoro-3-(trifluoromethyl)phenyl]-1-[5-(morpholin-4-yl)pentyl]urea
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one