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3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-[(2-fluorophenyl)methyl]piperidine-1-carboxamide
4-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-2-methylpyrimidine
methyl 3-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}amino)-4-methoxybenzoate
N-(2-methoxyethyl)-2-methyl-N-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
N-ethyl-N-(2-phenoxyethyl)-2,1-benzoxazole-3-carboxamide
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
(2S,4S)-4-[4-({[(4-chlorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-4-amine
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]ethan-1-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(propan-2-yl)piperidin-1-yl]methyl}piperidin-2-one
4-(4-methoxyphenyl)-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-4-oxobutanamide
N4,6-dimethyl-N4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
N-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]phenyl}-2-methylpropanamide
1-[4-(azetidin-1-ylmethyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]urea
(3S,4R)-N-(2-chlorophenyl)-3-acetamido-4-(4-methoxyphenyl)pyrrolidine-1-carboxamide
5-{[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-(4-methylphenyl)-5-(pyridin-4-yl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-3-azaspiro[5.5]undecan-9-amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
3-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-methyl-1H-indole
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidine-2-carboxamide
(5S,9aS,9bS)-5-(5-ethylfuran-2-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}benzoic acid
N-cyclohexyl-4-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)piperidine-1-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-butyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3-methylthiophen-2-yl)methyl]acetamide
2-(4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
N-(furan-3-ylmethyl)-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-(3-ethynylbenzoyl)-N-(3-fluorophenyl)piperidin-3-amine
7-(3-chlorophenyl)-4-(1H-imidazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
3-{5-[3-(pyrrolidine-1-sulfonyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
2-(2-{[(3-fluorophenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[2-(dimethylamino)ethyl]-9-(1H-indole-6-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-(3-phenylpropyl)-1,4-diazepane
2-(2-phenyl-1H-imidazol-1-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]ethan-1-one
2-(4-chloro-1H-pyrazol-1-yl)-1-[4-(3-fluorophenoxy)piperidin-1-yl]ethan-1-one
1-(2-methoxy-5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-cyclohexyl-3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-cyclopentyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-6-oxopiperidine-3-carboxamide
N,N-dimethyl-5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)pyridin-2-amine
1-cyclopentyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]piperidine-3-carboxamide
4-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]piperidin-1-yl}-6-ethyl-2-(pyrrolidin-1-yl)pyrimidine
N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-4-propylpyrimidine-5-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2,3,6-tetramethylquinoline-4-carboxamide
2-(2,5-dimethylphenoxy)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
2-(2-methyl-1,3-thiazol-4-yl)-5-(3-propoxypiperidine-1-carbonyl)pyrimidin-4-ol