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N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-[(3R,4S)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
ethyl 3-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]amino}-1-benzothiophene-2-carboxylate
(2S,4R)-4-amino-N-methyl-1-{2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}pyrrolidine-2-carboxamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
(1R,9aR)-1-[({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
4-(4-phenyl-1-{2-[(pyridin-3-yl)amino]ethyl}-1H-imidazol-5-yl)benzonitrile
[3-(3-{[4-(1H-imidazol-2-yl)piperidin-1-yl]methyl}phenoxy)propyl]dimethylamine
(3aS,6aS)-2-(1H-1,3-benzodiazol-2-ylmethyl)-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
[1-({methyl[(2,4,5-trimethylphenyl)methyl]amino}methyl)cyclopropyl]methanol
3-({cyclopropyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}methyl)phenol
2-amino-1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpropan-1-one
4-[2-(1H-pyrazol-1-yl)benzoyl]thiomorpholine
2,6-dimethyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]quinoline-4-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(cyclopropylmethyl)-N-propylacetamide
2-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-azaspiro[4.4]nonane
N-cyclooctyl-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyridin-4-amine
3-(3-{2-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)imidazolidine-2,4-dione
3-({2-[1-(3,4-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{2-[(3,5-dimethyl-1-benzofuran-2-yl)formamido]ethyl}pyridine-3-carboxamide
2-cyclopropyl-8-(heptan-4-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-{[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]methyl}-6-methylpyridin-3-ol
N-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)acetamide
1-[(2,4-difluoro-3-methoxyphenyl)methyl]piperidine-4-carbonitrile
3-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-(3-sulfamoylphenyl)urea
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidin-2-amine
(1R,2R,6S,7S)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(3aS,6aR)-5-{[2-(difluoromethoxy)phenyl]methyl}-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-cyclopentyl-3-[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
(4aS,8aS)-2-(2,6-dimethylpyridin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
N-[2-(dimethylsulfamoyl)ethyl]-2-(methylsulfanyl)pyrimidine-5-carboxamide
ethyl 1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
2-(1,4-dimethylpiperazin-2-yl)-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]acetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-(6-ethoxy-4-methylquinazolin-2-yl)azepan-4-amine
5-methyl-5-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
4-[3-(3-methoxypropyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(oxolan-2-ylmethyl)amino]pyridine-2-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
(4aS,8aS)-2-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-decahydroisoquinolin-4a-ol
1-[4-(2-phenoxyethyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
{4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]phenyl}methanol
2-[(3-methoxyphenyl)methyl]-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-[(dimethylamino)methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]azepan-4-ol
2-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
[1-(oxolane-3-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
(2R,3R)-3-(4-cyclohexylpiperazin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(3aR,5S,6S,7aS)-2-(2,3-dichlorobenzenesulfonyl)-octahydro-1H-isoindole-5,6-diol