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1-{4-[(5-ethylfuran-2-yl)methyl]piperazine-2-carbonyl}-4-methylpiperazine
1-cyclobutanecarbonyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
5-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoxaline
6-cyano-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]pyridine-3-carboxamide
(1R,5S,6R)-3-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(methylamino)pyridine-3-carboxamide
N-[4-(difluoromethoxy)-2-methylphenyl]-4-(pyridin-3-yl)piperazine-1-carboxamide
5-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carbonyl}-1-methyl-1H-1,3-benzodiazole
4-methyl-1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepan-5-one
(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-(propan-2-yloxy)phenyl)methanol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-(4-methoxyphenyl)-4-(4,4,4-trifluorobutyl)piperazine
4-methoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
5-(5-{[(4-methylphenyl)sulfanyl]methyl}furan-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(1-ethyl-1H-pyrazol-4-yl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carboxamide
N-methyl-N-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)methanesulfonamide
2-(1-{[1-(2,5-dimethylbenzenesulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-ethyl-8-{[3-(pyridin-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-(5-acetylthiophen-3-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
8-(butan-2-yl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(furan-2-yl)propanoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N3-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)piperidine-1,3-dicarboxamide
2-[3-(4-benzoylpiperazine-1-carbonyl)piperidin-1-yl]ethan-1-ol
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1-(9H-purin-6-yl)piperidin-4-amine
2-(4-methoxy-2,6-dimethylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
3-(dimethylamino)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
3-[4-(5-chlorofuran-2-carbonyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
4-(piperidin-1-ylmethyl)-N-[2-(pyridin-3-yloxy)propyl]benzamide
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N-(3-hydroxypropyl)-1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperidine-3-carboxamide
2-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}pyridine-4-carbonitrile
4-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}pyridine
2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-(thiophen-2-yl)-1,3-thiazole
N-benzyl-5-(1-methyl-1H-pyrazol-4-yl)furan-2-carboxamide
(1S,5R)-3-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-benzyl-3-[(cyclopent-3-en-1-yl)amino]-N-ethylpropanamide
N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)cyclopropanesulfonamide
8-(4-hydroxybenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(methylamino)ethan-1-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
5-methyl-1-propyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
2-(3-phenylpiperazin-1-yl)-4-(pyridin-3-yl)pyrimidine
(2S,3R)-3-hydroxy-2-[({[2-methyl-6-(propan-2-yl)phenyl]carbamoyl}methyl)amino]butanamide