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3-[(5-methyl-1H-imidazol-4-yl)methyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-[2-(dimethylamino)ethyl]-4-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-2-one
2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(4-fluorophenyl)ethan-1-ol
N-[3-({methyl[3-(oxolan-2-yl)propyl]carbamoyl}methoxy)phenyl]propanamide
3-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
N-(3-carbamoyl-4-methoxyphenyl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
2-[2-(1H-indazol-1-yl)phenyl]acetic acid
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-cyclohexyl-N-(prop-2-yn-1-yl)propanamide
3-{5-[2-(1H-imidazol-4-yl)-1-(1H-pyrrol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-(5-chloro-2-methoxyphenyl)-3-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
7-cyclohexyl-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-benzyl-5-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(dimethylamino)ethyl]-2-ethyl-N-[(5-methylthiophen-2-yl)methyl]pyrimidine-5-carboxamide
(1S,6R)-9-(2-ethoxypyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
N-[3-(methylsulfanyl)propyl]-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
2-(1-benzothiophen-2-yl)-4-[1-(furan-2-ylmethyl)pyrrolidin-3-yl]pyridine
4-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
4-ethyl-3-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5-[3-cyclopentyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
{1-[1-(4-methylquinazolin-2-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}(phenyl)methanol
methyl[(1-methyl-1H-imidazol-2-yl)methyl][(3-methylpyridin-2-yl)methyl]amine
4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}thiomorpholine
3-phenyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
7-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyrazolo[1,5-a]pyrimidine
(3aR,6aS)-2-{[4-(cyclopentyloxy)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-(3-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepine-2-carboxamide
3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[2-(piperidin-1-ylmethyl)phenyl]urea
2-(3-methyl-4-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-2-oxopiperazin-1-yl)acetic acid
ethyl 2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)acetate
3-methyl-1-propyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
3-(azocan-1-yl)-N-[1-(pyridin-4-yl)propan-2-yl]propanamide
N-(1,3-benzothiazol-2-ylmethyl)-N'-(2-fluoro-5-methylphenyl)butanediamide
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4-methylpyridine-3-carboxamide
N-(2-methoxyethyl)-2,5-dimethyl-N-[(2-methylphenyl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[5-(4-fluorophenyl)-1,3,4-thiadiazol-2-yl]-1-[2-(pyridin-3-yl)ethyl]urea
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
4-[3-(propoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
1-{3-[3-(2-methylpropyl)-1-phenyl-1H-1,2,4-triazol-5-yl]propyl}piperidin-2-one
4-[(3,5-difluorophenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[(1-benzylpiperidin-4-yl)methyl](1H-imidazol-4-ylmethyl)methylamine
5-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
N6-methyl-N6-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-9H-purine-2,6-diamine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(pyridin-3-yl)acetamide
N-cyclopentyl-2-(2-{[(2-methoxyethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)propanamide