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3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-4-[(2-methoxyphenyl)methyl]piperazin-2-one
2-{1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
1-(cyclohexylmethyl)-5-(4-formylpiperazin-1-yl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-hydroxyethyl)-4-[(1-methoxybutan-2-yl)amino]-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
dimethyl({[(1R,5S,6S)-3-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
2-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
3-(benzylamino)-N-[(4-methoxyphenyl)methyl]-5-(pyrrolidine-1-sulfonyl)benzamide
1'-(1-methyl-1H-pyrazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
(2S)-N-[(1-benzylpiperidin-4-yl)methyl]-2-hydroxy-N-methyl-2-phenylacetamide
N2-(1H-1,3-benzodiazol-2-ylmethyl)-N2,N4,N4,5-tetramethylpyrimidine-2,4-diamine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide
[2-(quinolin-8-yl)phenyl]methanol
dimethyl[(4-methyl-5-{1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-methylpiperidine
1-(2-amino-9H-purin-6-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
methyl 4-[4-(2-cyanobenzoyl)piperazin-1-yl]benzoate
N-cyclopropyl-1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-cyclopropyl-6-methoxy-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-acetyl-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
N,N-dimethyl-6-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]pyrimidin-4-amine
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[2-({[1-(2-carbamoylethyl)-1H-indol-3-yl]methyl}amino)ethyl]-2-chlorobenzamide
N-(2-methoxy-5-methylphenyl)-2-[(2-methyloxolan-2-yl)formamido]acetamide
2-(1-methyl-1H-pyrrol-3-yl)-N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]acetamide
2-{2-methyl-3-[({2-[(pyridin-3-yl)amino]ethyl}amino)methyl]-1H-indol-1-yl}acetamide
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
(4aS,7aR)-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2-methoxyethyl)-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,6R)-3-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
(5-{1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-(2-hydroxy-3-methoxypropyl)-N,4-dimethyl-6H,7H,8H-cyclopenta[g]quinazolin-2-amine
(3R,4S)-4-(propan-2-yl)-1-(propane-2-sulfonyl)pyrrolidin-3-amine
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-1H-pyrazole-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-[(3-fluorophenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazine
(2R,4S)-4-hydroxy-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine-2-carboxylic acid
3-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
[1-(1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}piperidin-4-yl)piperidin-3-yl]methanol
1-methyl-N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(carbamoylmethyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
8-[2-(3,4,5-trimethoxyphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(4S,6R)-6-methyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,4-diazepane-6-carboxylic acid