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1-cyclobutanecarbonyl-4-[(2,4,5-trimethylphenyl)methyl]-1,4-diazepane
2-[2-(trifluoromethyl)morpholin-4-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-({[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
1-(azocan-1-yl)-3-[5-methoxy-2-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-(4,4-difluoropiperidin-1-yl)-2-methyl-5-propylpyrimidine
1-[4-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)cyclohexyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-{5,6-dimethyl-4-[3-(piperidin-1-yl)azetidin-1-yl]thieno[2,3-d]pyrimidin-2-yl}ethan-1-amine
3-(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
1-[(2-chlorophenyl)methyl]-3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-6-methyl-1,2-dihydroquinolin-2-one
6-methoxy-2-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-(6-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}pyridin-2-yl)ethan-1-ol
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{[(4-methylphenyl)methyl]amino}benzamide
(3aS,6aS)-2-methyl-5-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,3S)-2-amino-1-(4-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-methylpentan-1-one
1-[2-methoxy-5-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-[2-(4-fluorophenyl)ethyl]-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(thiophene-3-carbonyl)piperidin-3-yl]piperazine
(2R,3R,6R)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4R)-4-(3-fluorophenyl)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
4-(3-hydroxyazetidin-1-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(2-methyl-1-benzofuran-7-yl)urea
1-(3,5-dimethylphenyl)-4-(quinolin-6-ylmethyl)piperazin-2-one
3-[5-(1H-imidazol-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidin-2-amine
(1S,2S,9R)-11-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
methyl 2-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-1H-1,3-benzodiazole-6-carboxylate
2-[2-(2-fluorophenyl)ethyl]-4-(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
(2S)-N1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyrrolidine-1,2-dicarboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-ethoxyphenyl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(2S,4S)-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-3-ylmethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{[(3,5-dimethylphenyl)methyl]sulfanyl}-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
2-(2-methoxyethyl)-N-(4-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-[(6-methoxypyrimidin-4-yl)amino]-N-methylethane-1-sulfonamide
N-cycloheptyl-1-cyclopropyl-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methyl}piperidin-4-ol
3-(4-methoxy-3,5-dimethylphenyl)-1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)urea
2-(3,5-dimethyl-1H-pyrazol-4-yl)-5-(pyrrolidin-1-ylmethyl)pyridine
2-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]benzoic acid
6-amino-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-3-carboxamide
5-methyl-3-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amine
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide