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3-[(3R,4S)-4-(dimethylamino)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propanoic acid
3-(4-methanesulfonylphenyl)-1-methyl-1-[1-(pyridin-3-yl)pentyl]urea
5-(cyclopentylamino)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
(1S,5R)-6-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
(3S,4R)-1-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]thiophene-2-carboxylic acid
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[4-(adamantan-1-yl)piperazine-1-carbonyl]-5-methylpyrazine
N-[2-(1H-indol-3-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
3-(2-aminoethyl)-4-(2,3-dimethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopentyl-5-(methoxymethyl)-N-(3-phenylprop-2-yn-1-yl)furan-2-carboxamide
3-(2-ethoxyethyl)-2-oxo-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
3-(1-hydroxybutan-2-yl)-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-methyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
1-[1-(4-hydroxy-4-methylpentan-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-3-(2-methanesulfonylethyl)urea
1-{1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]pyrrolidin-3-yl}-1H-imidazole
4-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-methylphenol
5-propyl-4-{4-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]piperidin-1-yl}pyrimidine
1-ethyl-4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperazin-2-one
1-(3-methoxybenzoyl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
N-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)-N-(prop-2-en-1-yl)butanamide
1-{5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
2-{4-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}pyrimidine
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidine-4-carbonitrile
(3R,4R)-4-ethyl-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidine-3,4-diol
N-{3-[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
5-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
7-chloro-2-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}-3-methyl-1H-indole
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(1S,5R)-6-(3,5-difluorobenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(2-fluorophenyl)methyl](2-methoxyethyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
methyl 6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidine-4-carboxylate
8-fluoro-2-[4-(pyrazin-2-yl)piperazine-1-carbonyl]quinoline
4-(5-chloro-2-methylphenyl)-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(methoxymethyl)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)cyclobutane-1-carboxamide
4-{[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}pyridine
4-(2-butoxyacetyl)-1-phenylpiperazin-2-one
8-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]acetamide
1-(3-fluorophenyl)-3-{1-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea