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4-[(1-ethylpyrrolidin-2-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
3-{1-[3-hydroxy-1-(4-methylphenyl)propyl]-1H-1,2,3-triazol-4-yl}benzonitrile
5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclohexylmethyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[N-benzyl-3-(1,2-oxazinan-2-yl)propanamido]acetic acid
propyl N-{[(2S,4S)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}carbamate
N-[2-(oxane-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-4-(trifluoromethyl)benzamide
(1S,4S)-2-(2-chlorophenyl)-5-(2,3-dihydro-1H-inden-2-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-ethyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4S)-4-[4-({[(2,4-difluorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
5-(1-methanesulfonylpyrrolidin-2-yl)-1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazole
{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
N-(1-methoxypropan-2-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
{1-[(5-fluoro-2-methoxyphenyl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
5-[(2-butylpyrrolidin-1-yl)methyl]-2-hydroxybenzoic acid
5-{2-[4-(3-methylphenyl)piperazin-1-yl]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
2-[1-(3-fluoro-4-methylbenzoyl)pyrrolidin-3-yl]benzoic acid
N-(2-methoxyethyl)-4-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
7-[(3-methoxyphenyl)methyl]-2-(3-methyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
N-(4-{1-[1-(thiophen-2-yl)propyl]-1H-imidazol-2-yl}phenyl)acetamide
2-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-8-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N3-[(3-fluorophenyl)methyl]-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxo-N-phenylacetamide
4-chloro-3-({[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]carbamoyl}amino)-N-methylbenzamide
1-tert-butyl-3-[2-(methylsulfanyl)ethyl]-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
4-{[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
3-{2-[2-(4-fluorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
1-methyl-4-[2-(methylsulfanyl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-chloro-3-ethyl-4-[(3-methoxypyrrolidin-1-yl)methyl]-1-methyl-1H-pyrazole
1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide
3-{[4-methoxy-4-(prop-2-en-1-yl)piperidin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
N-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-3-phenyl-1H-pyrazole-4-carboxamide
4-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperidine-4-carbonyl)morpholine
2-(3-methoxyphenyl)-N-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]azetidine-1-carboxamide
N-(oxan-4-yl)-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(pyridin-2-yl)acetamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxylic acid
N-[3-(3-methylphenyl)phenyl]-1-propanoylpiperidine-3-carboxamide
N-methyl-N-(oxan-4-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
4-fluoro-N-[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]benzamide