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(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-ol
6-(2-chlorophenyl)-2-(4-{[ethyl(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(1H-indol-5-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
4-(1,2-oxazol-5-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}thiophene-2-sulfonamide
8-(dimethyl-1,3-thiazole-5-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2,6-dimethylphenoxy)ethyl]-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
6-[2-(naphthalen-1-ylmethyl)morpholine-4-carbonyl]-2,3-dihydropyridazin-3-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[1-(dimethylamino)-2-methylpropan-2-yl]acetamide
2-(2-hydroxyethyl)-6-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
(4aR,7aS)-1-(2-methylpropyl)-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[3-(methylsulfanyl)propyl]propanamide
4-benzyl-3-(piperidin-4-yl)-1-[2-(pyrrolidin-1-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (2S,4S)-4-{[(2-ethylphenyl)carbamoyl]formamido}-1-methylpyrrolidine-2-carboxylate
N-[(2-chlorophenyl)methyl]-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}propanamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
N-[2-(diethylamino)ethyl]-N'-(2,4-dimethylphenyl)-N-methylpropanediamide
2-methyl-9-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-N-(pyridin-4-ylmethyl)piperidin-4-amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3,4,5-trifluorobenzoyl)pyrrolidin-3-yl]methanol
2-[(3-methylpiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-4-(1H-imidazol-1-yl)benzamide
3-[1-(5-ethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
8-(1-benzofuran-2-ylmethyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-ethyl-4-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1H-pyrazole-5-carboxamide
5-{1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-[4-(pyridin-3-yloxy)phenyl]urea
1-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
(3ar,6ar)-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-hydroxy-5-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)benzoic acid
4-[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]pyrimidine-5-carboxylic acid
N-(2-{1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
4-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-1-(4-methoxyphenyl)piperazin-2-one
(2S,4S,5R)-4-(azepane-1-carbonyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3,3,3-trifluoropropan-1-one
(2S)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylpiperidine-2-carboxamide
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-[4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)phenoxy]pyrimidine
6-cyclopentyl-N-[1-(furan-2-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-(1-benzofuran-5-ylmethyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-(1-benzoylpiperidin-4-yl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
N3-benzyl-N5-(1-benzylpiperidin-4-yl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,5-dimethylphenoxy)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-(4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
N-(2-methylpropyl)-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-N-(thiophen-3-ylmethyl)propanamide
N-[5-(4-phenyl-1H-imidazol-1-yl)pyridin-2-yl]methanesulfonamide
1-tert-butyl-5-[2-(4-methoxyphenyl)ethyl]-3-methyl-1H-1,2,4-triazole
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-[3-fluoro-5-(propan-2-yloxy)phenyl]-N,N-dimethylpyridine-3-carboxamide
(3R,4S)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-cyclopropylpyrrolidin-3-amine