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8-fluoro-2-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
[1-(2-phenoxyethanesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-(2-fluoro-4-methylphenyl)-2-[(4-methylpentan-2-yl)amino]acetamide
3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrrolidine
9-(cyclopropylmethyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
8-[(3-fluoro-2-methylphenyl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(1-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}ethyl)dimethylamine
1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperidine-3-carboxylic acid
1-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-(2-methoxyethyl)-1-methylurea
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}isoquinoline
1-[(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
1-(4-chlorobenzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
5-{[benzyl(methyl)amino]methyl}-N,N-diethyl-1,2-oxazole-3-carboxamide
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]quinoline-4-carboxylic acid
2-[(4-chlorophenyl)methyl]-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
2-cyclopentyl-N-(1H-imidazol-2-ylmethyl)-2-phenylacetamide
3-{[cyclohexyl(methyl)amino]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-(4-methoxyphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}oxan-4-amine
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyrrolidin-1-yl)ethan-1-one
(1S,5R)-6-(furan-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S)-1-{5-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
2,4-dimethyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)pyrimidine-5-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-pyrazol-1-yl]acetamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-(furan-3-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]quinoline-6-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(4-methyl-1H-imidazole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aR,7aS)-1-methyl-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(2-fluorophenyl)formamido]-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-methyl-5-(propan-2-yl)-N-[1-(pyridin-3-yl)pentyl]-1,2-oxazole-3-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-(pyridazine-4-carbonyl)piperazin-2-one
3-{6-amino-5-cyano-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridin-2-yl}benzoic acid
2-hydroxy-5-{1-[4-methoxy-3-(methylcarbamoyl)phenyl]-1H-imidazol-2-yl}benzoic acid
N-[2-(dimethylamino)ethyl]-3-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}propanamide
N-[2-(ethylsulfanyl)ethyl]-8-methylimidazo[1,2-a]pyridine-2-carboxamide
3-(3-methoxypropyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxylic acid
2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]pyridine-4-carboxamide
1-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-3-propylurea
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-phenyl-1H-pyrazole-5-carboxamide
1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
2,6-dimethoxy-4-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
(3aR,6aR)-2-(2-methoxyethyl)-5-(9H-purin-6-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-methoxyethyl)-8-{[3-(propan-2-yloxy)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N,3,5,7-tetramethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-indole-2-carboxamide
N2-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine